SCHEMBL27282920

SCHEMBL27282920

Cc1ccc(-c2c(C(N)=O)cc(-c3cnn(C)c3)n2COCC[Si](C)(C)C)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.41
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
RRM1 P23921 1/20 0.35
RRM2B Q7LG56 1/20 0.35
MKNK1 Q9BUB5 2/20 0.35
MKNK2 Q9HBH9 2/20 0.35
AXL P30530 1/20 0.35
MERTK Q12866 1/20 0.35
MAPK1 P28482 1/20 0.35
NPC1 O15118 1/20 0.35
KIT P10721 1/20 0.34
ALOX5AP P20292 2/20 0.34
FEN1 P39748 2/20 0.34
HCRTR1 O43613 4/20 0.34
GRM2 Q14416 2/20 0.34
MET P08581 2/20 0.34
PDK2 Q15119 1/20 0.33
ROCK2 O75116 1/20 0.33
HCRTR2 O43614 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27282917 0.85 NPC1 (0.35) NPC1ALOX5APFEN1GRM2ROCK2
SCHEMBL27282901 0.83 BAZ2B (0.38) ALOX5APFEN1
SCHEMBL27282921 0.81 NPC1 (0.35) NPC1ALOX5APFEN1GRM2
SCHEMBL27282919 0.80 NPC1 (0.35) BTKMKNK1MKNK2NPC1GRM2
SCHEMBL27282923 0.77 NUDT1 (0.39) NPC1MET
SCHEMBL16336797 0.74 MKNK1 (0.39) BTKMKNK1MKNK2NPC1GRM2
SCHEMBL27082828 0.69 ROCK2 (0.39) NPC1ROCK2
SCHEMBL27282698 0.69 MAPK14 (0.40) HCRTR1METHCRTR2
SCHEMBL27282898 0.69 ROCK2 (0.35) ALOX5APFEN1ROCK2
SCHEMBL27082584 0.68 BTK (0.57) BTKMKNK1MKNK2MAPK1PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240217969-A1 SUBSTITUTED PYRROLE CARBOXAMIDES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2024-07-04 US disclosed
US-20240217969-A1 SUBSTITUTED PYRROLE CARBOXAMIDES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2024-07-04 US disclosed
CN-117157289-A Substituted pyrrolecarboxamides, process for their preparation and their use as kinase inhibitors 内尔维亚诺医疗科学公司 2023-12-01 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240217969-A1 SUBSTITUTED PYRROLE CARBOXAMIDES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS KINASE INHIBITORS CDC7, CDK7, CDK17 BTK 488/4885CHRM2 4665/4885CHRM1 4555/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.