SCHEMBL2728338

SCHEMBL2728338

Cc1c(C(N)=O)cc(-c2cnccn2)c(C)c1-c1nccs1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.37
CYP3A4 P08684 2/20 0.34
CYP2C9 P11712 1/20 0.34
PKMYT1 Q99640 1/20 0.34
SIRT3 Q9NTG7 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
ADORA3 P0DMS8 1/20 0.33
TSHR P16473 1/20 0.33
MC4R P32245 1/20 0.33
ADRA1A P35348 1/20 0.33
MC3R P41968 1/20 0.33
CDC7 O00311 1/20 0.33
DBF4 Q9UBU7 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
TYK2 P29597 1/20 0.33
MAPK8 P45983 1/20 0.32
MAPK9 P45984 1/20 0.32
MAPK10 P53779 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2729192 0.85 CHEK2 (0.40) CHEK2CYP3A4CYP2C9PKMYT1TYK2
SCHEMBL2728017 0.84 NPSR1 (0.42) CHEK2CDC7KDM4EALDH1A1SCN9A
SCHEMBL2726268 0.77 CFTR (0.37) CHEK2CYP3A4CYP2C9PKMYT1TYK2
SCHEMBL2726309 0.72 CYP3A4 (0.42) CHEK2CYP3A4CYP2C9PKMYT1SIRT3
SCHEMBL1932926 0.71 CHEK2 (0.38) CHEK2CYP3A4CYP2C9PKMYT1TDP1
SCHEMBL3350408 0.71 SMPD3 (0.46) CHEK2CYP3A4CYP2C9PKMYT1HDAC1
SCHEMBL28531660 0.70 SIRT3 (0.36) PKMYT1SIRT3TDP1ADORA3TSHR
SCHEMBL2728335 0.69 TGFBR1 (0.42) CYP3A4CYP2C9PKMYT1ADORA3TSHR
SCHEMBL27983939 0.68 CHEK2 (0.39) CHEK2CYP3A4CYP2C9PKMYT1ADORA3
SCHEMBL27986525 0.67 CHEK2 (0.45) CHEK2SIRT3TDP1ADORA3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed