SCHEMBL2729192

SCHEMBL2729192

Cc1c(C(N)=O)cc(-c2nccs2)c(C)c1-c1nccs1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.40
TYK2 P29597 1/20 0.36
EEF2K O00418 2/20 0.35
TUBB4A P04350 2/20 0.35
TUBB P07437 2/20 0.35
TUBA3C P0DPH7 2/20 0.35
TUBA1B P68363 2/20 0.35
TUBA4A P68366 2/20 0.35
TUBB4B P68371 2/20 0.35
TUBB3 Q13509 2/20 0.35
TUBB2A Q13885 2/20 0.35
TUBB8 Q3ZCM7 2/20 0.35
TUBA3E Q6PEY2 2/20 0.35
TUBA1A Q71U36 2/20 0.35
TUBA1C Q9BQE3 2/20 0.35
TUBB6 Q9BUF5 2/20 0.35
TUBB2B Q9BVA1 2/20 0.35
TUBB1 Q9H4B7 2/20 0.35
LRRK2 Q5S007 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2728017 0.85 NPSR1 (0.42) CHEK2PTGDR2ALDH1A1SCN9ARAB9A
SCHEMBL2728338 0.85 CHEK2 (0.37) CHEK2TYK2CYP3A4CYP2C9PKMYT1
SCHEMBL2726268 0.85 CFTR (0.37) CHEK2TYK2EEF2KTUBB4ATUBB
SCHEMBL2726309 0.79 CYP3A4 (0.42) CHEK2EEF2KLRRK2CYP3A4CYP2C9
SCHEMBL1932926 0.79 CHEK2 (0.38) CHEK2TYK2EEF2KLRRK2CYP3A4
SCHEMBL3350408 0.79 SMPD3 (0.46) CHEK2LRRK2CYP3A4CYP2C9PKMYT1
SCHEMBL27983939 0.78 CHEK2 (0.39) CHEK2TYK2CYP3A4CYP2C9PKMYT1
SCHEMBL2733045 0.75 TYK2 (0.43) CHEK2TYK2TUBB4ATUBBTUBA3C
SCHEMBL30810277 0.74 CHEK2 (0.40) CHEK2TYK2TUBB4ATUBBTUBA3C
SCHEMBL30810232 0.74 ACLY (0.37) CHEK2TYK2EEF2KLRRK2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed