SCHEMBL2729191

SCHEMBL2729191

Cc1csc(-c2cc(-c3nccs3)cc(C(N)=O)c2C)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.43
TGFBR1 P36897 2/20 0.39
SPHK2 Q9NRA0 1/20 0.38
SPHK1 Q9NYA1 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
SMPD3 Q9NY59 1/20 0.37
PIK3CB P42338 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
S100A4 P26447 1/20 0.36
LRRK2 Q5S007 1/20 0.35
PLAU P00749 1/20 0.35
MYC P01106 1/20 0.35
PKMYT1 Q99640 1/20 0.34
F2 P00734 1/20 0.34
F10 P00742 1/20 0.34
PLG P00747 1/20 0.34
F7 P08709 1/20 0.34
F3 P13726 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2729187 0.84 CHEK2 (0.37) CHEK2TGFBR1SPHK2SPHK1SMPD3
SCHEMBL3350408 0.84 SMPD3 (0.46) CHEK2PTGDR2SMPD3PIK3CBLRRK2
SCHEMBL2728335 0.80 TGFBR1 (0.42) TGFBR1PIK3CBNPC1RAB9AS100A4
SCHEMBL2728014 0.80 PDE10A (0.54) CHEK2TGFBR1RAB9AEIF4E
SCHEMBL2726265 0.80 TGFBR1 (0.38) TGFBR1PIK3CBNPC1RAB9ASMN1; SMN2
SCHEMBL2729192 0.74 CHEK2 (0.40) CHEK2PTGDR2SMPD3RAB9ASMN1; SMN2
SCHEMBL1932926 0.73 CHEK2 (0.38) CHEK2TGFBR1PTGDR2SMPD3PIK3CB
SCHEMBL3347230 0.73 CHEK2 (0.41) CHEK2PTGDR2SMPD3NPC1RAB9A
SCHEMBL1933814 0.72 CHEK2 (0.41) CHEK2TGFBR1SPHK2SPHK1PIK3CB
SCHEMBL2726308 0.71 TGFBR1 (0.46) TGFBR1NPC1RAB9ASMN1; SMN2S100A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed