SCHEMBL2729449

SCHEMBL2729449

COC(=O)[C@H](Cc1ccc(O[Si](C)(C)C(C)(C)CCCCl)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.50
ITGA2B P08514 2/20 0.50
KLK5 Q9Y337 1/20 0.45
HDAC8 Q9BY41 1/20 0.42
PTPN1 P18031 2/20 0.42
YAP1 P46937 1/20 0.41
CTSS P25774 6/20 0.41
CTSK P43235 5/20 0.41
BCL2 P10415 1/20 0.41
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
KMT2A Q03164 1/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
ACE P12821 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20437145 0.85 ITGB3 (0.52) ITGB3ITGA2BKLK5HDAC8PTPN1
SCHEMBL2729447 0.84 ITGB3 (0.48) ITGB3ITGA2BKLK5HDAC8PTPN1
SCHEMBL2728593 0.81 ITGB3 (0.60) ITGB3ITGA2BKLK5HDAC8PTPN1
SCHEMBL5892285 0.81 ITGB3 (0.60) ITGB3ITGA2BKLK5HDAC8PTPN1
SCHEMBL14365476 0.81 ITGB3 (0.56) ITGB3ITGA2BKLK5HDAC8PTPN1
SCHEMBL16173545 0.81 ITGB3 (0.56) ITGB3ITGA2BKLK5HDAC8PTPN1
SCHEMBL5408855 0.78 PPARG (0.57) ITGB3ITGA2BKLK5HDAC8CTSS
SCHEMBL5408845 0.78 PPARG (0.57) ITGB3ITGA2BKLK5HDAC8CTSS
SCHEMBL8232330 0.78 ITGB3 (0.62) ITGB3ITGA2BKLK5HDAC8PTPN1
SCHEMBL12056445 0.78 ITGB3 (0.59) ITGB3ITGA2BKLK5HDAC8PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012058325-A1 COMPOUNDS AND METHODS USEFUL FOR TREATMENT OF DISEASES MEDIATED BY HIF-1 ONCOTHYREON INC. (US) 2012-05-03 WO disclosed