SCHEMBL27304547

SCHEMBL27304547

N#Cc1ccc(NCc2ccccc2F)nc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN2 Q96KS0 1/20 0.50
MAP4K4 O95819 1/20 0.48
IDH1 O75874 3/20 0.47
LRRK2 Q5S007 1/20 0.45
VNN1 O95497 2/20 0.43
NPC1 O15118 1/20 0.43
PKM P14618 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
NTRK1 P04629 1/20 0.41
NTRK3 Q16288 1/20 0.41
NTRK2 Q16620 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
ALDH1A1 P00352 3/20 0.40
CYP1A2 P05177 3/20 0.40
CYP2C19 P33261 3/20 0.40
CYP2C9 P11712 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL507660 0.79 NTRK1 (0.56) EGLN2VNN1SMN1; SMN2MEN1KMT2A
SCHEMBL1882080 0.78 SMN1; SMN2 (0.68) MAP4K4VNN1NPC1PKMRAB9A
SCHEMBL1267858 0.77 CYP3A4 (0.55) EGLN2NTRK3CYP2C19CYP2C9CYP3A4
SCHEMBL32683749 0.77 IDH1 (0.44) IDH1VNN1MEN1KMT2ANTRK1
SCHEMBL27304831 0.75 NPC1 (0.58) IDH1NPC1PKMRAB9ASMN1; SMN2
SCHEMBL1882774 0.75 VNN1 (0.47) MAP4K4VNN1NPC1PKMRAB9A
SCHEMBL27304412 0.75 NTRK1 (0.61) EGLN2MAP4K4LRRK2VNN1NTRK1
SCHEMBL27302479 0.75 MEN1 (0.54) SMN1; SMN2MEN1KMT2AMAPTL3MBTL1
SCHEMBL6638863 0.74 DPP4 (0.53) IDH1MEN1KMT2AALDH1A1CYP1A2
SCHEMBL29580404 0.73 ALDH1A1 (0.65) MAP4K4NPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024029489-A1 KIT INHIBITORS, COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE THEREOF MODULUS DISCOVERY, INC. (JP) 2024-02-08 WO disclosed