SCHEMBL27315136

SCHEMBL27315136

CC(=O)c1[nH]c2ccc(O)c(F)c2c1Br

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NEK1 Q96PY6 1/20 0.34
GPR35 Q9HC97 1/20 0.34
MAP2 P11137 2/20 0.33
ERN1 O75460 1/20 0.31
MTNR1A P48039 1/20 0.30
MTNR1B P49286 1/20 0.30
PRNP P04156 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
PPARG P37231 1/20 0.30
HIF1A Q16665 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30
NR2E3 Q9Y5X4 1/20 0.30
NCOR2 Q9Y618 1/20 0.30
MET P08581 1/20 0.30
EIF4A3 P38919 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27302892 0.76 FEN1 (0.43) MTNR1AMTNR1B
SCHEMBL12228580 0.68 MAP2 (0.46) MAP2CYP1A2CYP2C9CYP2C19NPSR1
SCHEMBL16065345 0.67 PDE3B (0.38) ERN1CYP1A2CYP2C9CYP2C19MET
SCHEMBL23000274 0.65 MAP2 (0.40) MAP2CYP1A2CYP2C9CYP2C19NPSR1
SCHEMBL21884849 0.65 AR (0.36) MAP2ERN1NPSR1MET
SCHEMBL28424735 0.65 KDM4E (0.49) MAP2
SCHEMBL5324128 0.64 BRD4 (0.36) ERN1RXFP1
SCHEMBL2462946 0.64 KDM4E (0.51) CYP1A2CYP2C9CYP2C19NPSR1
SCHEMBL8371524 0.61 RXFP1 (0.54) MAP2PRNPCYP1A2CYP2C9CYP2C19
SCHEMBL12255399 0.61 EGFR (0.39) MTNR1AMTNR1BCYP1A2CYP2C19NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1031222-A β-(fluorine methylene radical)-5-hydroxytryptophan and derivative as the monoamine oxidase prodrugs for inhibition MERRELL DOW PHARMA (US) 1989-02-22 CN claimed