SCHEMBL21884849

SCHEMBL21884849

Cc1[nH]c2ccc(O)c(F)c2c1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.36
DAO P14920 1/20 0.36
MET P08581 1/20 0.35
ERN1 O75460 1/20 0.35
CYP17A1 P05093 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
MEN1 O00255 4/20 0.34
KMT2A Q03164 4/20 0.34
ALDH1A1 P00352 4/20 0.34
MAPT P10636 4/20 0.34
HPGD P15428 4/20 0.34
GAA P10253 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
CDK1 P06493 1/20 0.32
CDK2 P24941 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16065345 0.85 PDE3B (0.38) DAOMETERN1HTR2AHTR2C
SCHEMBL2462946 0.73 KDM4E (0.51) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL5324128 0.73 BRD4 (0.36) ERN1MEN1KMT2AALDH1A1MAPT
SCHEMBL12255399 0.70 EGFR (0.39) MEN1KMT2AALDH1A1MAPTGAA
SCHEMBL16065320 0.68 GPR84 (0.38) ERN1HTR2AHTR2CESR1ESR2
SCHEMBL13127020 0.67 CYP3A4 (0.37) CYP17A1CYP11B1CYP11B2KMT2AALDH1A1
SCHEMBL12620997 0.67 MAP2 (0.39) MAP2
SCHEMBL27315136 0.65 NEK1 (0.34) METERN1NPSR1MAP2
SCHEMBL3426211 0.64 DAO (0.55) ARDAOALDH1A1MAPTCDK2
SCHEMBL296024 0.64 KEAP1 (0.47) DAOMEN1KMT2AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112996784-B Indole derivatives and their use in medicine 北京越之康泰生物医药科技有限公司 2023-05-30 CN disclosed
CN-112996784-A Indole derivatives and their use in medicine 北京越之康泰生物医药科技有限公司 2021-06-18 CN disclosed
WO-2020057403-A1 INDOLE DERIVATIVE AND MEDICAL APPLICATION THEREOF 北京越之康泰生物医药科技有限公司 2020-03-26 WO disclosed