SCHEMBL2731679

SCHEMBL2731679

COc1cc(OC(C)=O)ccc1-n1cnnn1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.57
TSHR P16473 2/20 0.57
KMT2A Q03164 2/20 0.50
HPGD P15428 2/20 0.50
NPSR1 Q6W5P4 1/20 0.48
PKM P14618 3/20 0.48
LMNA P02545 2/20 0.48
USP2 O75604 1/20 0.47
HSD17B10 Q99714 1/20 0.47
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2731444 0.83 KMT2A (0.45) ALDH1A1TSHRKMT2AHPGDPKM
SCHEMBL2732579 0.83 KMT2A (0.45) ALDH1A1TSHRKMT2AHPGDPKM
SCHEMBL2730327 0.79 KMT2A (0.67) ALDH1A1TSHRKMT2AHPGDPKM
SCHEMBL2731678 0.75 KMT2A (0.54) ALDH1A1TSHRKMT2ANPSR1PKM
SCHEMBL15825106 0.75 KMT2A (0.71) KMT2ALMNAUSP2
SCHEMBL2729430 0.74 KCNJ1 (0.65) ALDH1A1TSHRKMT2AHPGDPKM
SCHEMBL4580901 0.73 ALDH1A1 (0.49) ALDH1A1TSHRKMT2AHPGDNPSR1
SCHEMBL15018034 0.73 KCNJ1 (0.49) ALDH1A1TSHRKMT2AHPGD
SCHEMBL17232502 0.72 ALDH1A1 (0.67) ALDH1A1TSHRKMT2APKMLMNA
SCHEMBL153056 0.71 CA12 (0.59) ALDH1A1TSHRKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2632464-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL Merck Sharp & Dohme Corp. (US) 2013-09-04 EP disclosed
WO-2012058134-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME CORP. (US) 2012-05-03 WO disclosed