SCHEMBL27318

SCHEMBL27318

CCCCCCNC(=O)OC1(O)CC[C@@]2(C)C(=CC[C@H]3[C@@H]4CC[C@H]([C@H](C)CCCC(C)C)[C@@]4(C)CC[C@@H]32)C1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP46A1 Q9Y6A2 2/20 0.56
USP2 O75604 2/20 0.56
LMNA P02545 1/20 0.56
ABCB1 P08183 1/20 0.56
OSBP P22059 1/20 0.56
RORC P51449 1/20 0.56
OSBP2 Q969R2 1/20 0.56
POLA1 P09884 1/20 0.56
GRIN1 Q05586 14/20 0.54
GRIN2B Q13224 14/20 0.54
GRIN2A Q12879 12/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4654756 0.89 USP2 (0.59) CYP46A1USP2LMNAABCB1OSBP
SCHEMBL18797660 0.87 USP2 (0.58) CYP46A1USP2LMNAABCB1OSBP
SCHEMBL10929500 0.86 USP2 (0.65) CYP46A1USP2LMNAABCB1OSBP
SCHEMBL10930823 0.86 USP2 (0.65) CYP46A1USP2LMNAABCB1OSBP
SCHEMBL10929495 0.86 USP2 (0.65) CYP46A1USP2LMNAABCB1OSBP
SCHEMBL16926435 0.85 CYP46A1 (0.69) CYP46A1USP2LMNAABCB1OSBP
SCHEMBL17129625 0.85 CYP46A1 (0.69) CYP46A1USP2LMNAABCB1OSBP
SCHEMBL10622619 0.85 CYP46A1 (0.69) CYP46A1USP2LMNAABCB1OSBP
SCHEMBL20470662 0.85 CYP46A1 (0.69) CYP46A1USP2LMNAABCB1OSBP
SCHEMBL16299806 0.85 CYP46A1 (0.69) CYP46A1USP2LMNAABCB1OSBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 10520 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250313818-A1 CRISPR-Cas Effector Polypeptides and Methods of Use Thereof THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2025-10-09 US claimed
US-12215343-B2 Methods and compositions for RNA-directed target DNA modification and for RNA-directed modulation of transcription THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-02-04 US claimed
EP-3419665-B1 TREATMENT METHODS FOR FIBROSIS TARGETING SMOC2 BRIGHAM & WOMENS HOSPITAL INC (US) 2024-10-30 EP claimed
US-12123015-B2 Methods and compositions for RNA-directed target DNA modification and for RNA-directed modulation of transcription THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-10-22 US claimed
US-20240229029-A9 COMPOSITIONS AND METHODS FOR TREATMENT OF FRIEDREICH'S ATAXIA THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2024-07-11 US claimed
US-20240141348-A1 ALLELE SELECTIVE INHIBITION OF MUTANT C9ORF72 FOCI EXPRESSION BY DUPLEX RNAS TARGETING THE EXPANDED HEXANUCLEOTIDE REPEAT THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2024-05-02 US claimed
US-11970711-B2 Methods and compositions for RNA-directed target DNA modification and for RNA-directed modulation of transcription THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-04-30 US claimed
US-20240132889-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF FRIEDREICH'S ATAXIA THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2024-04-25 US claimed
WO-2023201203-A2 CRISPR-CAS EFFECTOR POLYPEPTIDES AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-10-19 WO claimed
US-11674159-B2 Methods and compositions for RNA-directed target DNA modification and for RNA-directed modulation of transcription THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-06-13 US claimed
US-20020039741-A1 Antitumor agent DEAN NICHOLAS M (US) 2002-04-04 US claimed
EP-0957926-A4 OLIGONUCLEOTIDE COMPOSITIONS AND METHODS FOR THE MODULATION OF THE EXPRESSION OF B7 PROTEIN ISIS PHARMACEUTICALS INC (US) 2002-01-23 EP claimed
US-6319906-B1 FOR THERAPY OF AUTOIMMUNE DISEASE, INFLAMMATORY DISEASE, FOR INHIBITING ALLOGRAFT REJECTION ISIS PHARMACEUTICALS 2001-11-20 US claimed
US-6312900-B1 FOR MODULATING METASTASIS OF MALIGNANT TUMORS VIA MODULATION OF ACTIVATING PROTEIN 1 ISIS PHARMACEUTICALS, INC. 2001-11-06 US claimed
JP-2000507833-A 2000-06-27 JP claimed
US-6077833-A FOR DIAGNOSIS, PREVENTION AND TREATMENT OF IMMUNE STATES AND DISORDERS AMENABLE TO TREATMENT THROUGH MODULATION OF T CELL ACTIVATION SUCH AS FOR PREVENTING ALLOGRAFT REJECTION ISIS PHARMACEUTICALS, INC. (US) 2000-06-20 US claimed
US-6001991-A NUCLEOTIDE SEQUENCES WHICH HYBRIDIZE TO AND SUPPRESS EXPRESSION OF MULTIDRUG RESISTANCE GENE; FOR PREVENTING OR MODULATING THE DEVELOPMENT OF MULTIDRUG RESISTANCE DURING CHEMOTHERAPEUTIC TREATMENT OR RESENSITIZING TREATED CELLS ISIS PHARMACEUTICALS INC. (US) 1999-12-14 US claimed
EP-0957926-A1 OLIGONUCLEOTIDE COMPOSITIONS AND METHODS FOR THE MODULATION OF THE EXPRESSION OF B7 PROTEIN ISIS PHARMACEUTICALS, INC. (US) 1999-11-24 EP claimed
WO-1998029124-A1 OLIGONUCLEOTIDE COMPOSITIONS AND METHODS FOR THE MODULATION OF THE EXPRESSION OF B7 PROTEIN ISIS PHARMACEUTICALS, INC. (US) 1998-07-09 WO claimed
WO-1998014615-A1 ANTISENSE OLIGONUCLEOTIDE MODULATION OF MDR P-GLYCOPROTEIN GENE EXPRESSION ISIS PHARMACEUTICALS, INC. (US) 1998-04-09 WO claimed