SCHEMBL27319829

SCHEMBL27319829

Cc1cc(O)c2scc(C(=O)O)c2n1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EIF4EBP1 Q13541 11/20 0.38
KDM4E B2RXH2 1/20 0.36
CSNK2A1 P68400 1/20 0.36
GPR35 Q9HC97 2/20 0.36
LCK P06239 1/20 0.35
SORT1 Q99523 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19554455 0.85 ALDH1A1 (0.42) EIF4EBP1KDM4EGPR35LCKSORT1
SCHEMBL22866767 0.83 KDM4E (0.40) KDM4E
SCHEMBL29560113 0.83 KDM4E (0.40) KDM4E
SCHEMBL28715107 0.83 GPR35 (0.45) EIF4EBP1KDM4EGPR35SORT1
SCHEMBL28704856 0.83 EIF4EBP1 (0.41) EIF4EBP1
SCHEMBL28704402 0.79 EIF4EBP1 (0.54) EIF4EBP1
SCHEMBL22866890 0.78 HPGD (0.37) KDM4EGPR35
SCHEMBL19698920 0.73 GPR35 (0.41) EIF4EBP1KDM4EGPR35
SCHEMBL28717584 0.71 GPR35 (0.38) KDM4EGPR35
SCHEMBL29560349 0.70 PARP1 (0.39) KDM4ESORT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024103067-A1 COMPOUNDS AND COMPOSITIONS AS eIF4E INHIBITORS AND USES THEREOF RIBOMETRIX, INC. (US) 2024-05-16 WO disclosed
CN-114269756-B 4-Oxo-3, 4-dihydropyrido [3,4-D ] pyrimidine compounds that inhibit EIF4E 效应疗法股份有限公司 2024-05-14 CN disclosed
CN-114269756-A 4-oxo-3, 4-dihydropyrido [3,4-D ] pyrimidine compounds inhibiting EIF4E 效应疗法股份有限公司 2022-04-01 CN disclosed