SCHEMBL2732045

SCHEMBL2732045

CS(=O)(=O)c1c(CC(=O)O)ccc2c1COC2=O

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 14/20 0.41
KCNH2 Q12809 7/20 0.41
AKR1B1 P15121 2/20 0.40
ACHE P22303 1/20 0.36
SSTR1 P30872 1/20 0.36
SLC6A4 P31645 1/20 0.36
PTGS2 P35354 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL286817 0.80 KCNJ1 (0.58) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL30751813 0.80 KCNJ1 (0.58) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL299969 0.80 KCNJ1 (0.44) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL300175 0.77 KCNJ1 (0.43) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL9517001 0.75 AKR1B1 (0.43) KCNJ1KCNH2AKR1B1PTGS2
SCHEMBL300308 0.75 KCNJ1 (0.41) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL3808243 0.74 KCNJ1 (0.43) KCNJ1KCNH2ACHESSTR1SLC6A4
Hydrochloric Acid SCHEMBL2733903 0.71 KCNJ1 (0.57) KCNJ1KCNH2
SCHEMBL14921946 0.70 KCNJ1 (0.50) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL300145 0.69 KCNJ1 (0.40) KCNJ1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2632465-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL Merck Sharp & Dohme Corp. (US) 2013-09-04 EP disclosed
WO-2012058116-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME CORP. (US) 2012-05-03 WO disclosed