SCHEMBL2732938

SCHEMBL2732938

CC1(C(F)(F)F)COC(=O)N1c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 3/20 0.36
ALDH1A1 P00352 2/20 0.36
ATM Q13315 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
IDH1 O75874 7/20 0.35
CACNA1B Q00975 1/20 0.34
APBA1 Q02410 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8475478 0.74 IDH1 (0.51) HSD11B1ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL8475475 0.74 IDH1 (0.51) HSD11B1ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL3570167 0.70 IDH1 (0.38) HSD11B1ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL3576644 0.69 HSD11B1 (0.37) HSD11B1ALDH1A1ATMCYP1A2CYP2C9
SCHEMBL20340441 0.68 IDH1 (0.46) HSD11B1ALDH1A1ATMIDH1SMN1; SMN2
SCHEMBL5418053 0.66 IDH1 (0.38) ALDH1A1ATMIDH1
SCHEMBL17149455 0.66 TSHR (0.46) ALDH1A1CYP1A2CYP2C9CYP2C19IDH1
Hydrochloric Acid SCHEMBL17140395 0.65 TSHR (0.45) ALDH1A1CYP1A2CYP2C9CYP2C19IDH1
SCHEMBL7812799 0.65 ALDH1A1 (0.35) HSD11B1ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL8475165 0.65 GAA (0.36) HSD11B1ALDH1A1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143193-B Biaryl or heterocyclic biaryl substituted cyclohexene derivative compounds as CETP inhibitors 株式会社钟根堂 2017-12-15 CN disclosed
EP-2632269-A1 CYCLIC AMINE SUBSTITUTED OXAZOLIDINONE CETP INHIBITOR Merck Sharp & Dohme Corp. (US) 2013-09-04 EP disclosed
WO-2012058187-A1 CYCLIC AMINE SUBSTITUTED OXAZOLIDINONE CETP INHIBITOR MERCK SHARP & DOHME CORP. (US) 2012-05-03 WO disclosed