SCHEMBL27336255

SCHEMBL27336255

C[Si](C)(C)CCOCn1ccc2c(C(F)(F)F)c[nH]c(=O)c21

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 3/20 0.38
DUT P33316 1/20 0.36
EGFR P00533 1/20 0.33
IGF1R P08069 1/20 0.33
SRC P12931 1/20 0.33
FLT4 P35916 1/20 0.33
KDR P35968 1/20 0.33
FLT3 P36888 1/20 0.33
EPHB4 P54760 1/20 0.33
TEK Q02763 1/20 0.33
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL32667111 0.83 DUT (0.36) DGAT1DUTEGFRIGF1RSRC
SCHEMBL30902997 0.82 DUT (0.35) DGAT1DUTEGFRIGF1RSRC
SCHEMBL30728198 0.79 DUT (0.35) DGAT1DUTEGFRIGF1RSRC
SCHEMBL31319360 0.76 NPC1 (0.32) NPC1
SCHEMBL30903046 0.76 DGAT1 (0.43) DGAT1EGFRIGF1RSRCFLT4
SCHEMBL31319438 0.75 DGAT1 (0.35) DGAT1
SCHEMBL31319343 0.74 PDE3B (0.32)
SCHEMBL27041330 0.73 DUT (0.37) DGAT1DUTEGFRIGF1RSRC
SCHEMBL6719621 0.72 DGAT1 (0.42) DGAT1DUTEGFRIGF1RSRC
SCHEMBL30479870 0.72 MAPT (0.42) DGAT1DUTEGFRIGF1RSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024105563-A1 SUBSTITUTED BICYCLIC PYRIDONE DERIVATIVES PFIZER INC. (US) 2024-05-23 WO disclosed
WO-2024105563-A1 SUBSTITUTED BICYCLIC PYRIDONE DERIVATIVES PFIZER INC. (US) 2024-05-23 WO disclosed