SCHEMBL27337208

SCHEMBL27337208

c1ccc(-c2ccc(N(c3ccccc3-c3cccc4c3ccc3c5ccccc5oc43)c3cccc4ccccc34)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 3/20 0.40
PRKDC P78527 4/20 0.33
GGPS1 O95749 1/20 0.33
CYP1A1 P04798 4/20 0.33
CYP1A2 P05177 4/20 0.33
CYP1B1 Q16678 4/20 0.33
MAPT P10636 4/20 0.33
ABCG2 Q9UNQ0 3/20 0.33
KDM4E B2RXH2 3/20 0.33
ALDH1A1 P00352 3/20 0.33
HPGD P15428 3/20 0.33
HSD17B10 Q99714 3/20 0.33
ABCC1 P33527 2/20 0.33
TP53 P04637 2/20 0.33
TSHR P16473 2/20 0.33
MAPK1 P28482 2/20 0.33
PDE5A O76074 1/20 0.33
ABCB1 P08183 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23233344 0.94 ALOX5 (0.43) ALOX5PRKDCGGPS1MAPTKDM4E
SCHEMBL27336959 0.93 ALOX5 (0.41) ALOX5PRKDCGGPS1CYP1A1CYP1A2
SCHEMBL27337207 0.93 ALOX5 (0.41) ALOX5PRKDCGGPS1CYP1A1CYP1A2
SCHEMBL27337403 0.93 ALOX5 (0.40) ALOX5PRKDCGGPS1MAPTKDM4E
SCHEMBL24471763 0.93 ALOX5 (0.40) ALOX5PRKDCGGPS1MAPTKDM4E
SCHEMBL24825406 0.92 ALOX5 (0.39) ALOX5PRKDCGGPS1CYP1A1CYP1A2
SCHEMBL24889046 0.92 ALOX5 (0.39) ALOX5PRKDCGGPS1CYP1A1CYP1A2
SCHEMBL27337186 0.92 ALOX5 (0.39) ALOX5PRKDCGGPS1CYP1A1CYP1A2
SCHEMBL27336941 0.92 ALOX5 (0.39) ALOX5PRKDCGGPS1CYP1A1CYP1A2
SCHEMBL27297063 0.92 ALOX5 (0.39) ALOX5PRKDCGGPS1CYP1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023199832-A1 COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENTS, ORGANIC ELECTROLUMINESCENT ELEMENT, AND ELECTRONIC DEVICE 出光興産株式会社 2023-10-19 WO disclosed