SCHEMBL27353259

SCHEMBL27353259

Cn1c(=O)sc2cc(CCC(N)Cc3ccc(C(F)(F)F)cc3)ccc21

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.52
SIGMAR1 Q99720 11/20 0.47
HTR2C P28335 4/20 0.43
AKT1 P31749 2/20 0.42
CDK2 P24941 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27353257 0.76 AKT1 (0.59) HTR1AHTR2CAKT1CDK2
SCHEMBL8948338 0.76 HTR1A (0.54) HTR1ASIGMAR1HTR2C
Hydrochloric Acid SCHEMBL8871795 0.72 SIGMAR1 (0.57) HTR1ASIGMAR1HTR2C
SCHEMBL9685737 0.71 SIGMAR1 (0.64) HTR1ASIGMAR1HTR2C
SCHEMBL7761420 0.70 SIGMAR1 (0.59) HTR1ASIGMAR1HTR2C
SCHEMBL8114163 0.70 SIGMAR1 (0.61) HTR1ASIGMAR1HTR2C
SCHEMBL4614132 0.69 EPHX1 (0.50) HTR2CAKT1CDK2
Hydrochloric Acid SCHEMBL8870817 0.69 SIGMAR1 (0.60) HTR1ASIGMAR1HTR2C
SCHEMBL9684012 0.68 MAPT (0.61) HTR1ASIGMAR1HTR2C
SCHEMBL9484568 0.68 SIGMAR1 (0.62) HTR1ASIGMAR1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1050601-C Preparation and the pharmaceutical compositions which contain them ADIR (FR) 2000-03-22 CN disclosed
CN-1111626-A Preparation and the pharmaceutical compositions which contain them ADIR (FR) 1995-11-15 CN disclosed