SCHEMBL27363041

SCHEMBL27363041

COc1ccc(N)c(-c2nnn[nH]2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.42
CYP3A4 P08684 4/20 0.42
GAA P10253 2/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
GFER P55789 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
MAPT P10636 4/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
THRB P10828 2/20 0.39
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
NPC1 O15118 2/20 0.38
KDM4E B2RXH2 2/20 0.38
RECQL P46063 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11360946 0.88 ALDH1A1 (0.42) ALDH1A1CYP3A4GAAMAPK1HTT
SCHEMBL16549277 0.79 AMY1A (0.42) ALDH1A1GAAMAPK1HTTGFER
SCHEMBL9132775 0.79 SLC6A2 (0.42) ALDH1A1CYP3A4GAAMAPK1HTT
SCHEMBL4326211 0.78 HSP90AA1 (0.44) ALDH1A1CYP3A4GAAMAPK1HTT
SCHEMBL11361203 0.78 HSD17B10 (0.36) ALDH1A1CYP3A4GAAMAPK1HTT
SCHEMBL20329381 0.76 ALDH1A1 (0.37) ALDH1A1CYP3A4GAAMAPK1HTT
SCHEMBL9132682 0.76 SLC6A2 (0.47) ALDH1A1CYP3A4GAAMAPK1HTT
SCHEMBL9134917 0.76 SLC6A2 (0.49) ALDH1A1CYP3A4GAAMAPK1HTT
SCHEMBL17914525 0.76 TEK (0.37) ALDH1A1GAAMAPK1HTTGFER
SCHEMBL20329237 0.76 MAPT (0.44) ALDH1A1CYP3A4GAAMAPK1GFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1073089-C Benzodiazepine derivatives, compositions thereof and their use in the manufacture of medicaments SHIONOGI & CO (JP) 2001-10-17 CN disclosed
CN-1143362-A Novel benzodizaepine derivative SHIONOGI & CO (JP) 1997-02-19 CN disclosed