SCHEMBL27363663

SCHEMBL27363663

COc1cc2[nH]nc(C(=O)O)c2cc1OC

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKAA1 Q13131 14/20 0.57
PRKAG1 P54619 13/20 0.57
PRKAB1 Q9Y478 13/20 0.57
PRKAB2 O43741 12/20 0.54
PRKAA2 P54646 12/20 0.54
PRKAG3 Q9UGI9 12/20 0.54
PRKAG2 Q9UGJ0 12/20 0.54
TLR8 Q9NR97 2/20 0.44
TLR7 Q9NYK1 2/20 0.44
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
DYRK3 O43781 1/20 0.43
MAP4K4 O95819 1/20 0.43
CDK1 P06493 1/20 0.43
CDK2 P24941 1/20 0.43
MARK3 P27448 1/20 0.43
CLK2 P49760 1/20 0.43
GSK3B P49841 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27777072 0.89 PRKAG1 (0.47) PRKAA1PRKAG1PRKAB1PRKAB2PRKAA2
SCHEMBL1963808 0.88 PRKAG1 (0.53) PRKAA1PRKAG1PRKAB1PRKAB2PRKAA2
SCHEMBL1963540 0.88 PRKAG1 (0.53) PRKAA1PRKAG1PRKAB1PRKAB2PRKAA2
SCHEMBL12479871 0.87 KDM4E (0.44) PRKAA1PRKAG1PRKAB1PRKAB2PRKAA2
SCHEMBL1964504 0.83 PRKAG1 (0.48) PRKAA1PRKAG1PRKAB1PRKAB2PRKAA2
SCHEMBL14915843 0.82 PRKAG1 (0.46) PRKAA1PRKAG1PRKAB1PRKAB2PRKAA2
SCHEMBL10569944 0.81 KDM4E (0.58) PRKAA1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL7809574 0.80 KDM4E (0.59) KDM4EALDH1A1HPGDSMN1; SMN2GAA
SCHEMBL13931932 0.79 TUBB1 (0.46)
SCHEMBL13632234 0.79 PRKAG1 (0.53) PRKAA1PRKAG1PRKAB1PRKAB2PRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1067998-C Hydrate for medicinal use DAIICHI PHARMACEUDTICAL CO LTD (JP) 2001-07-04 CN disclosed
CN-1171786-A Hydrate for medicinal use DAIICHI SEIYAKU CO (JP) 1998-01-28 CN disclosed
CN-1100301-A Drug for neuroprotection DAIICHI SEIYAKU CO (JP) 1995-03-22 CN disclosed