SCHEMBL27366096

SCHEMBL27366096

O=C1C=C2Oc3ccccc3N=C2C(=O)C1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
HRH4 Q9H3N8 1/20 0.31
RARA P10276 1/20 0.30
RARB P10826 1/20 0.30
RXRA P19793 1/20 0.30
RXRB P28702 1/20 0.30
RXRG P48443 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28386848 0.81 CYP1A2 (0.30) CYP1A2CYP2D6HDAC3HDAC1HDAC2
SCHEMBL7007833 0.70 MAPT (0.38) KDM4EALDH1A1LMNAGAAMAPT
Hydrochloric Acid SCHEMBL7004514 0.69 MAPT (0.37) KDM4EALDH1A1LMNAGAAMAPT
Hydrochloric Acid SCHEMBL7004542 0.69 MAPT (0.37) KDM4EALDH1A1LMNAGAAMAPT
SCHEMBL7451103 0.69 CA12 (0.39) LMNA
SCHEMBL11818614 0.68 HDAC6 (0.33) KDM4ENPC1ALDH1A1MAPTRAB9A
SCHEMBL30960181 0.66 PKM (0.32) KDM4E
SCHEMBL15549945 0.65 KDM4E (0.36) CYP1A2CYP2D6KDM4ENPC1ALDH1A1
SCHEMBL7002550 0.63 ALDH1A1 (0.38) KDM4ENPC1ALDH1A1LMNAMAPT
SCHEMBL4083532 0.62 ALDH1A1 (0.40) CYP1A2CYP2D6KDM4ENPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1067686-C Fused polycyclic heterocycle derivatives EISAI CO LTD (JP) 2001-06-27 CN disclosed
CN-1185781-A Fused Polycyclic Heterocyclic Derivatives EISAI CO LTD (JP) 1998-06-24 CN disclosed