SCHEMBL27366264

SCHEMBL27366264

CCCOn1c(=O)c2c(ncn2Cc2ccccc2)n(CC(C)C)c1=O

nearest known ligand 0.69

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE1A P54750 5/20 0.69
PDE1B Q01064 5/20 0.69
PDE1C Q14123 5/20 0.69
SMN1; SMN2 Q16637 3/20 0.50
ALDH1A1 P00352 2/20 0.50
ADORA2B P29275 1/20 0.50
RXFP1 Q9HBX9 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
PDE2A O00408 4/20 0.49
POLB P06746 1/20 0.48
HIF1A Q16665 1/20 0.48
KMT2A Q03164 4/20 0.46
CNOT7 Q9UIV1 3/20 0.45
MEN1 O00255 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7606356 0.85 PDE1A (0.67) PDE1APDE1BPDE1CSMN1; SMN2ALDH1A1
SCHEMBL1944565 0.84 PDE1A (0.82) PDE1APDE1BPDE1CSMN1; SMN2ALDH1A1
SCHEMBL1944712 0.74 POLB (0.70) PDE1APDE1BPDE1CSMN1; SMN2ALDH1A1
SCHEMBL7608527 0.74 POLB (0.59) PDE1APDE1BPDE1CSMN1; SMN2ALDH1A1
SCHEMBL7605727 0.74 KMT2A (0.55) PDE1APDE1BPDE1CSMN1; SMN2ALDH1A1
SCHEMBL7605036 0.74 BRD4 (0.68) PDE1APDE1BPDE1CSMN1; SMN2ALDH1A1
SCHEMBL555093 0.73 ALDH1A1 (0.65) PDE1APDE1BPDE1CSMN1; SMN2ALDH1A1
SCHEMBL1946890 0.72 POLB (0.67) PDE1APDE1BPDE1CSMN1; SMN2ALDH1A1
SCHEMBL3615415 0.71 ALDH1A1 (0.63) PDE1APDE1BPDE1CSMN1; SMN2ALDH1A1
SCHEMBL1947176 0.71 KMT2A (0.71) PDE1APDE1BPDE1CSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1066146-C Use of theophylline derivatives for curing and preventing shock state, xanthine derivatives and preparation thereof AVENTIS PHARMACEUTICALS AG (DE) 2001-05-23 CN disclosed
CN-1169993-A Use of theophylline derivatives for curing and preventing shock state, xanthine derivatives and preparation thereof HOECHST AG (DE) 1998-01-14 CN disclosed