SCHEMBL27380577

SCHEMBL27380577

COc1ccc(Cl)c(-c2ccc3c(=O)n(-c4cncc5ccccc45)c(=O)[nH]c3c2)c1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.42
PKM P14618 1/20 0.42
KDM4E B2RXH2 4/20 0.40
HPGD P15428 3/20 0.40
ALDH1A1 P00352 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
HIF1A Q16665 1/20 0.40
TP53 P04637 4/20 0.39
MEN1 O00255 1/20 0.38
ALOX12 P18054 1/20 0.38
KMT2A Q03164 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HTT P42858 1/20 0.38
MAPT P10636 2/20 0.36
NPEPPS P55786 1/20 0.36
EGLN3 Q9H6Z9 1/20 0.36
GRIA1 P42261 1/20 0.36
CACNG8 Q8WXS5 1/20 0.36
GAA P10253 1/20 0.35
ERN1 O75460 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27377882 0.89 GRIA1 (0.48) HSD17B10PKMKDM4EHPGDALDH1A1
SCHEMBL27378008 0.85 HSD17B10 (0.44) HSD17B10PKMKDM4EHPGDALDH1A1
SCHEMBL27380409 0.85 HSD17B10 (0.42) HSD17B10PKMKDM4EHPGDALDH1A1
SCHEMBL27192346 0.85 KDM4E (0.46) KDM4ETP53HTTNPEPPSGRIA1
SCHEMBL27379932 0.84 HSD17B10 (0.45) HSD17B10PKMKDM4EHPGDALDH1A1
SCHEMBL27191759 0.84 PTGES (0.46) KDM4ETP53HTTNPEPPSGAA
SCHEMBL27380562 0.83 HPGD (0.46) HSD17B10PKMKDM4EHPGDALDH1A1
SCHEMBL27378570 0.83 NPEPPS (0.39) HSD17B10PKMKDM4EHPGDALDH1A1
SCHEMBL27378372 0.82 HSD17B10 (0.45) HSD17B10PKMKDM4EHPGDALDH1A1
SCHEMBL27192042 0.82 HSD17B10 (0.48) HSD17B10PKMKDM4EHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024031089-A1 SARS-COV2 MAIN PROTEASE INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-08 WO disclosed