SCHEMBL2738809

SCHEMBL2738809

CN(CCOC(C)(c1ccccc1)c1ccc(Cl)cc1)P(=O)(O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 3/20 0.49
HTR1A P08908 2/20 0.49
ADRA2A P08913 2/20 0.49
CHRM1 P11229 2/20 0.49
DRD1 P21728 2/20 0.49
SLC6A2 P23975 2/20 0.49
SLC6A4 P31645 2/20 0.49
ADRA1A P35348 2/20 0.49
OPRM1 P35372 2/20 0.49
DRD3 P35462 2/20 0.49
SLC6A3 Q01959 2/20 0.49
KCNH2 Q12809 2/20 0.49
HRH3 Q9Y5N1 2/20 0.49
TBXA2R P21731 1/20 0.49
ACHE P22303 1/20 0.49
CYP3A4 P08684 2/20 0.48
CYP2D6 P10635 2/20 0.48
TMEM97 Q5BJF2 2/20 0.48
SIGMAR1 Q99720 2/20 0.48
SLC22A1 O15245 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2738810 0.89 CHRM2 (0.46) CHRM2HTR1AADRA2ACHRM1DRD1
SCHEMBL2738814 0.87 CHRM2 (0.47) CHRM2HTR1AADRA2ACHRM1DRD1
SCHEMBL2738811 0.86 CHRM2 (0.48) CHRM2HTR1AADRA2ACHRM1DRD1
SCHEMBL218014 0.84 CHRM2 (0.46) CHRM2HTR1AADRA2ACHRM1DRD1
Chlorphenoxamine SCHEMBL29208 0.82 CHRM2 (0.61) CHRM2HTR1AADRA2ACHRM1DRD1
SCHEMBL2738813 0.81 CHRM2 (0.46) CHRM2HTR1AADRA2ACHRM1DRD1
Chlorphenoxamine SCHEMBL125112 0.81 CHRM2 (0.59) CHRM2HTR1AADRA2ACHRM1DRD1
SCHEMBL2738882 0.80 CHRM2 (0.70) CHRM2CHRM1KCNH2CYP3A4CYP2D6
Chlorphenoxamine SCHEMBL1649036 0.80 CHRM2 (0.62) CHRM2HTR1AADRA2ACHRM1DRD1
Clofenetamine SCHEMBL2110100 0.77 CHRM2 (0.54) CHRM2HTR1AADRA2ACHRM1DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088918-B2 Noncardiotoxic pharmaceutical compounds WILLIAMSBURG HOLDINGS LLC (US) 2012-01-03 US disclosed
US-8088918-B2 Noncardiotoxic pharmaceutical compounds WILLIAMSBURG HOLDINGS LLC (US) 2012-01-03 US disclosed