SCHEMBL27403244

SCHEMBL27403244

COc1ccc(CNc2nc(Cl)nc3sccc23)cc1OC

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TNF P01375 1/20 0.68
NOD1 Q9Y239 1/20 0.68
NPC1 O15118 1/20 0.54
GALR3 O60755 1/20 0.54
LMNA P02545 1/20 0.54
NR2F2 P24468 1/20 0.54
HTT P42858 1/20 0.54
RAB9A P51151 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
APP P05067 7/20 0.51
ACHE P22303 7/20 0.49
BCHE P06276 4/20 0.49
STAT1 P42224 1/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
PDE5A O76074 1/20 0.47
GAA P10253 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27377633 0.92 TNF (0.57) TNFNOD1NPC1GALR3LMNA
SCHEMBL5128515 0.84 APP (0.51) TNFNOD1NPC1RAB9AAPP
SCHEMBL5128296 0.83 NPC1 (0.53) TNFNOD1NPC1GALR3NR2F2
SCHEMBL27655477 0.82 TNF (0.44) TNFNOD1RAB9AAPPPDE5A
SCHEMBL7404118 0.81 TNF (1.00) TNFNOD1NPC1GALR3LMNA
SCHEMBL5123734 0.81 APP (0.48) TNFNOD1NPC1RAB9AAPP
SCHEMBL5123492 0.80 ESR1 (0.67) TNFNOD1APPSTAT1PDE5A
SCHEMBL5120111 0.79 ACHE (0.47) TNFNOD1NPC1RAB9AAPP
SCHEMBL3121034 0.79 APP (0.79) APPACHEBCHESTAT1MEN1
Hydrochloric Acid SCHEMBL3123789 0.78 APP (0.77) APPACHEBCHESTAT1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1875023-A Use of thienopyrimidines MERCK PATENT GMBH (DE) 2006-12-06 CN disclosed
CN-1081638-C Thienopyrimidine compounds MERCK PATENT GMBH (DE) 2002-03-27 CN disclosed
CN-1227560-A Thienopyrimidines MERCK PATENT GMBH (DE) 1999-09-01 CN disclosed