SCHEMBL27425865

SCHEMBL27425865

Nc1cc(Cl)ccc1-c1ccncn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK10 P53779 1/20 0.47
MAPK14 Q16539 1/20 0.47
JAK2 O60674 1/20 0.41
TSHR P16473 2/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP3A4 P08684 2/20 0.41
ALOX15 P16050 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
MAP4K4 O95819 2/20 0.40
EGFR P00533 2/20 0.40
FRK P42685 2/20 0.40
MAPK9 P45984 2/20 0.40
SLK Q9H2G2 2/20 0.40
DCLK1 O15075 1/20 0.40
PRKD3 O94806 1/20 0.40
PRKACA P17612 1/20 0.40
FLT3 P36888 1/20 0.40
CSNK1A1 P48729 1/20 0.40
GSK3B P49841 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3232479 0.82 MAPT (0.49) MAPK10MAPK14ALDH1A1SMN1; SMN2MAP4K4
SCHEMBL27581704 0.79 JAK2 (0.47) MAPK10MAPK14JAK2MAP4K4EGFR
SCHEMBL27426787 0.79 TYR (0.40) MAPK10MAPK14MAP4K4EGFRFRK
SCHEMBL30464793 0.79 MAP4K4 (0.49) MAPK10MAPK14JAK2ALDH1A1MAP4K4
SCHEMBL3091852 0.77 NPC1 (0.50) TSHRALDH1A1CYP3A4ALOX15SMN1; SMN2
SCHEMBL28290775 0.76 EGFR (0.43) MAPK10MAPK14JAK2TSHRALDH1A1
SCHEMBL29453704 0.76 JAK2 (0.47) MAPK10MAPK14JAK2TSHRALDH1A1
SCHEMBL22719341 0.76 JAK2 (0.47) MAPK10MAPK14JAK2TSHRALDH1A1
SCHEMBL27865549 0.74 MAPK14 (0.43) MAPK10MAPK14JAK2MAP4K4EGFR
SCHEMBL27591971 0.74 ALDH1A1 (0.46) MAPK10MAPK14ALDH1A1SMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1109675-C Aryl pyrimidine derivatives HOFFMANN LA ROCHE (CH) 2003-05-28 CN disclosed
CN-1223641-A Aryl pyrimidine derivatives HOFFMANN LA ROCHE (CH) 1999-07-21 CN disclosed