SCHEMBL28290775

SCHEMBL28290775

Nc1ccc(-c2ccncn2)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.43
MAP4K4 O95819 2/20 0.43
FRK P42685 2/20 0.43
MAPK9 P45984 2/20 0.43
CSNK1A1 P48729 2/20 0.43
DCLK1 O15075 1/20 0.43
PRKD3 O94806 1/20 0.43
PRKACA P17612 1/20 0.43
FLT3 P36888 1/20 0.43
GSK3B P49841 1/20 0.43
MINK1 Q8N4C8 1/20 0.43
SLK Q9H2G2 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
MAP4K5 Q9Y4K4 1/20 0.43
KDM4E B2RXH2 2/20 0.41
NPC1 O15118 2/20 0.41
MAPT P10636 2/20 0.41
RAB9A P51151 2/20 0.41
ALDH1A1 P00352 2/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3232479 0.82 MAPT (0.49) EGFRMAP4K4FRKMAPK9CSNK1A1
SCHEMBL5685355 0.81 HSP90AA1 (0.41) EGFRMAP4K4FRKMAPK9CSNK1A1
SCHEMBL27877944 0.79 NPC1 (0.46) EGFRMAP4K4FRKMAPK9CSNK1A1
SCHEMBL7085680 0.79 HSP90AA1 (0.42) EGFRMAP4K4FRKMAPK9CSNK1A1
SCHEMBL13549952 0.77 NPC1 (0.50) KDM4ENPC1MAPTRAB9AALDH1A1
SCHEMBL17292996 0.76 MAPT (0.56) MAP4K4FRKMAPK9CSNK1A1PRKD3
SCHEMBL27425865 0.76 MAPK10 (0.47) EGFRMAP4K4FRKMAPK9CSNK1A1
SCHEMBL2650530 0.76 MAP4K4 (0.43) EGFRMAP4K4FRKMAPK9CSNK1A1
SCHEMBL5243501 0.76 NPC1 (0.45) KDM4ENPC1MAPTRAB9AALDH1A1
SCHEMBL16370824 0.76 AAK1 (0.51) CLK4KDM4EMAPTALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110214136-A Pyrazole derivatives as MALT1 inhibitor 詹森药业有限公司 2019-09-06 CN disclosed
CN-106170489-B New Pyrazolopyrimidine derivative and its purposes as MALT1 inhibitor 诺华股份有限公司 2019-05-03 CN disclosed