SCHEMBL6958211

SCHEMBL6958211

CC(=O)C(Cc1ccc(F)cc1)c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.60
ESR2 Q92731 1/20 0.60
EPHX1 P07099 2/20 0.53
TDP1 Q9NUW8 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
CHRM1 P11229 5/20 0.47
UBE2N P61088 1/20 0.47
POLB P06746 1/20 0.46
PPARA Q07869 2/20 0.46
PPARD Q03181 1/20 0.46
PPARG P37231 1/20 0.45
PTPN1 P18031 1/20 0.45
PTGS1 P23219 1/20 0.44
PTGS2 P35354 1/20 0.44
ALDH1A1 P00352 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5272849 0.88 EPHX1 (0.67) ESR1ESR2EPHX1CHRM1UBE2N
SCHEMBL4664796 0.86 PPARA (0.56) EPHX1TDP1CYP3A4CYP2D6CYP2C9
SCHEMBL3371227 0.85 ESR1 (0.62) ESR1ESR2EPHX1CHRM1UBE2N
SCHEMBL6049128 0.85 ESR1 (0.83) ESR1ESR2EPHX1CHRM1UBE2N
SCHEMBL8672896 0.83 EPHX1 (0.53) EPHX1TDP1CYP3A4CYP2D6CYP2C9
SCHEMBL3371208 0.83 ESR1 (0.60) ESR1ESR2EPHX1CYP2D6CYP2C9
SCHEMBL28835702 0.83 EPHX1 (0.77) EPHX1TDP1CYP3A4CYP2D6CYP2C9
SCHEMBL22394854 0.83 ESR1 (0.63) ESR1ESR2EPHX1TDP1CYP3A4
SCHEMBL27991442 0.81 EPHX1 (0.58) EPHX1CHRM1UBE2NPPARAPPARG
SCHEMBL27426752 0.81 ESR1 (0.57) ESR1ESR2EPHX1CHRM1UBE2N

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0325130-B1 Substituted pyridines BAYER AG (DE) 2003-11-05 EP disclosed
US-5401746-A FOR INHIBITING CHOLESTEROL BIOSYNTHESIS AND HMG-COA REDUCTASE BAYER AKTIENGESELLSCHAFT (DE) 1995-03-28 US disclosed
US-5169857-A Anticholesterol agents BAYER AKTIENGESELLSCHAFT (DE) 1992-12-08 US disclosed
US-5006530-A Certain 7-[2,6-diisopropyl-4-phenyl-5-lower alkoxymethyl-pyrid-3-yl]-3,5-dihydroxy-6-enoates and derivatives useful for treating circulatory diseases BAYER AKTIENGESELLSCHAFT (DE) 1991-04-09 US disclosed
EP-0325130-A2 Substituted pyridines BAYER AG (DE) 1989-07-26 EP disclosed
EP-0300278-A2 Process for the preparation of 2-substituted pyrroles BAYER AG (DE) 1989-01-25 EP disclosed