SCHEMBL27437868

SCHEMBL27437868

O=CC1Nc2cc(Cl)c(C(O)CCN3CCC(Cc4ccc(F)cc4)CC3)cc2N1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 4/20 0.50
GRIN1 Q05586 2/20 0.47
GMNN O75496 1/20 0.47
TP53 P04637 1/20 0.47
CYP3A4 P08684 1/20 0.47
ALOX15 P16050 1/20 0.47
TSHR P16473 1/20 0.47
NFKB1 P19838 1/20 0.47
THPO P40225 1/20 0.47
MTOR P42345 1/20 0.47
BLM P54132 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
CCR3 P51677 2/20 0.42
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
ADRA1D P25100 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41
GRIN2A Q12879 1/20 0.41
GRIN2C Q14957 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27460820 0.91 GRIN2B (0.52) GRIN2BGRIN1GMNNTP53CYP3A4
SCHEMBL27459644 0.86 GRIN2B (0.62) GRIN2BGRIN1GMNNTP53CYP3A4
SCHEMBL8542871 0.81 GRIN2B (0.54) GRIN2BGRIN1GMNNTP53CYP3A4
SCHEMBL27391248 0.79 GRIN2B (0.56) GRIN2BGRIN1GMNNTP53CYP3A4
SCHEMBL27460009 0.74 GRIN2B (0.64) GRIN2BGRIN1GRIN2DGRIN3BGRIN2A
SCHEMBL27459289 0.74 GRIN2B (0.54) GRIN2BGRIN1GRIN2DGRIN3BGRIN2A
SCHEMBL8544030 0.73 GRIN2B (0.55) GRIN2BGRIN1GMNNTP53CYP3A4
SCHEMBL28964579 0.72 GRIN2B (0.44) GRIN2BCCR3OPRM1
SCHEMBL8892949 0.72 GRIN2B (0.71) GRIN2BGRIN1GMNNTP53CYP3A4
SCHEMBL8547312 0.72 MAOA (0.54) GRIN2BGRIN1GRIN2DGRIN3BADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1128762-A Benzyl piperidine derivatives MERCK PATENT GMBH (DE) 1996-08-14 CN disclosed