Formaldehyde

Formaldehyde

SCHEMBL27445163

C=O.CS(=O)(=O)N[C@@H](Cc1ccccc1)C(=O)OCCl.CS(=O)(=O)N[C@@H](Cc1ccccc1)C(=O)OCCl

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.52
CA12 O43570 2/20 0.50
CA7 P43166 2/20 0.50
CA9 Q16790 2/20 0.50
CA14 Q9ULX7 2/20 0.50
CA2 P00918 1/20 0.50
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
ITGB3 P05106 1/20 0.46
ITGA2B P08514 1/20 0.46
MMP2 P08253 6/20 0.46
MMP9 P14780 4/20 0.46
ADAMTS4 O75173 1/20 0.46
CTSL P07711 2/20 0.45
CTSS P25774 1/20 0.45
HTT P42858 1/20 0.44
ADAMTS5 Q9UNA0 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
PPARG P37231 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9819677 0.85 POLB (0.55) POLBCA12CA7CA9CA14
SCHEMBL20335114 0.85 POLB (0.55) POLBCA12CA7CA9CA14
SCHEMBL6435869 0.84 POLB (0.69) POLBCA12CA7CA9CA14
SCHEMBL6435872 0.84 POLB (0.69) POLBCA12CA7CA9CA14
SCHEMBL20334978 0.84 POLB (0.69) POLBCA12CA7CA9CA14
Formaldehyde SCHEMBL19474730 0.83 CTSL (0.64) POLBCA7CA2MMP2MMP9
SCHEMBL698062 0.82 MMP2 (0.63) POLBITGB3ITGA2BMMP2MMP9
SCHEMBL698061 0.82 MMP2 (0.63) POLBITGB3ITGA2BMMP2MMP9
Benzene SCHEMBL28198278 0.82 MMP2 (0.63) POLBITGB3ITGA2BMMP2MMP9
SCHEMBL6436714 0.82 MMP2 (0.63) POLBITGB3ITGA2BMMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1163466-C Substituted oxobutanoic acid derivatives as matrix metalloproteinase inhibitors 2004-08-25 CN disclosed
CN-1139570-C Inhibition of matrix metalloproteases by acetylene contg. compounds 拜尔公司 2004-02-25 CN disclosed
CN-1124255-C Inhibition of matrix metalloproteases by substituted phenethyl compounds BAYER AG (US) 2003-10-15 CN disclosed
CN-1119313-C Inhibition of matrix metalloproteinases by 2- (omega-aroylalkyl) -4-diaryl-4-oxobutanoic acid BAYER AG (US) 2003-08-27 CN disclosed
CN-1100748-C Inhibition of matrix metalloproteinases by 2-substituted-4- (4-substituted phenyl) -4-oxobutanoic acid BAYER AG (US) 2003-02-05 CN disclosed
CN-1234791-A Inhibition of matrix metalloproteases by 2-('omega'-aroylalkyl)-4-biaryl-oxobutyric acids BAYER AG (US) 1999-11-10 CN disclosed
CN-1225621-A Inhibition of matrix metalloproteinases by 2-substituted-4- (4-substituted phenyl) -4-oxobutanoic acid BAYER AG (US) 1999-08-11 CN disclosed
CN-1225620-A Substituted 4-arylbutanoic acid derivatives as matrix metalloproteinase inhibitors BAYER AG (US) 1999-08-11 CN disclosed
CN-1225624-A Inhibition of matrix metalloproteases by substituted phenethyl compounds BAYER AG (US) 1999-08-11 CN disclosed
CN-1225622-A Substituted oxobutyric acids as matrix metalloprotease inhibitor BAYER AG (US) 1999-08-11 CN disclosed
CN-1225623-A Inhibition of matrix metalloproteases by acetylene contg. compounds BAYER AG (US) 1999-08-11 CN disclosed