SCHEMBL27449031

SCHEMBL27449031

Cc1ncccc1Oc1ccccc1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.49
PTGS2 P35354 2/20 0.49
SLC6A2 P23975 5/20 0.48
SLC6A4 P31645 4/20 0.48
SLC6A3 Q01959 4/20 0.48
HTR1A P08908 2/20 0.48
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
ADORA2A P29274 1/20 0.46
ADORA1 P30542 1/20 0.46
LMNA P02545 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HTT P42858 1/20 0.44
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
CCR2 P41597 1/20 0.42
CCR4 P51679 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6545410 0.86 ADORA2A (0.50) ADORA2AADORA1NPC1ALDH1A1CYP3A4
SCHEMBL28302902 0.83 S1PR4 (0.52) PTGS1PTGS2SLC6A2SLC6A4SLC6A3
SCHEMBL11881284 0.82 ADORA2A (0.45) ADORA2AADORA1CYP3A4CYP2C9CYP2C19
SCHEMBL11543918 0.81 SLC6A2 (0.47) PTGS1PTGS2SLC6A2SLC6A4SLC6A3
SCHEMBL4797448 0.80 GRM2 (0.42) PTGS1PTGS2SLC6A2SLC6A4HTR1A
SCHEMBL4797458 0.80 ADORA2A (0.43) SLC6A2SLC6A4HTR1AKMT2AMEN1
SCHEMBL2657071 0.78 NPC1 (0.50) SLC6A2SLC6A4SLC6A3HTR1AKMT2A
SCHEMBL2084341 0.77 ADORA2A (0.51) PTGS1PTGS2SLC6A2SLC6A4ADORA2A
SCHEMBL1436765 0.77 HPGD (0.59) PTGS1PTGS2SLC6A2SLC6A4SLC6A3
SCHEMBL9340516 0.76 NR1I2 (0.46) PTGS1PTGS2SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024138040-A1 METHODS OF TREATMENT WITH TRADIPITANT VANDA PHARMACEUTICALS INC. (US) 2024-06-27 WO disclosed