SCHEMBL27465716

SCHEMBL27465716

CS(=O)(=O)c1c(-c2ccccc2)ncc(Cl)c1N

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 3/20 0.42
LMNA P02545 2/20 0.42
HPGD P15428 2/20 0.42
GLA P06280 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 2/20 0.41
PTGS2 P35354 5/20 0.38
PTGS1 P23219 3/20 0.38
ADORA2A P29274 2/20 0.38
ADORA1 P30542 2/20 0.37
ATR Q13535 1/20 0.36
GAA P10253 1/20 0.35
LOXL3 P58215 1/20 0.35
LOXL2 Q9Y4K0 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5210203 0.78 LMNA (0.41) L3MBTL1ALDH1A1KDM4ELMNANPSR1
SCHEMBL27482775 0.77 PTGS2 (0.45) L3MBTL1LMNANPSR1PTGS2PTGS1
SCHEMBL27481298 0.76 PTGS2 (0.48) L3MBTL1ALDH1A1KDM4ELMNAHPGD
SCHEMBL27462731 0.73 PTGS2 (0.50) L3MBTL1LMNANPSR1PTGS2PTGS1
SCHEMBL28066 0.72 PTGS2 (0.48) L3MBTL1LMNANPSR1PTGS2PTGS1
Hydrochloric Acid SCHEMBL27483154 0.72 PTGS2 (0.49) L3MBTL1LMNANPSR1PTGS2PTGS1
SCHEMBL27548124 0.72 KDM4E (0.41) L3MBTL1ALDH1A1KDM4ELMNAHPGD
Hydrochloric Acid SCHEMBL27468627 0.72 PTGS2 (0.47) L3MBTL1LMNANPSR1PTGS2PTGS1
SCHEMBL5207597 0.71 PTGS2 (0.40) L3MBTL1ALDH1A1KDM4ELMNANPSR1
SCHEMBL27482777 0.71 PTGS2 (0.47) L3MBTL1LMNANPSR1PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1152863-C Substituted pyridines as selective cyclooxygenase-2 inhibitors ��˸���˹��(���ô�)��˾ 2004-06-09 CN disclosed
CN-1225085-A Substituted pyridines as selective cyclooxygenase-2 inhibitors MERCK FROSST CANADA INC (CA) 1999-08-04 CN disclosed