Hydroxycamptothecin

Hydroxycamptothecin

SCHEMBL27466705

CCC1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3cc(O)ccc3nc2-1.[NaH]

nearest known ligand 0.98

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 18/20 0.98
MEN1 O00255 4/20 0.98
KMT2A Q03164 4/20 0.98
SMN1; SMN2 Q16637 4/20 0.98
ALDH1A1 P00352 4/20 0.98
KDM4E B2RXH2 3/20 0.98
CYP3A4 P08684 2/20 0.98
HBB P68871 2/20 0.98
CASP1 P29466 1/20 0.98
CASP7 P55210 1/20 0.98
GLA P06280 3/20 0.79
TP53 P04637 2/20 0.79
HPGD P15428 2/20 0.79
STAT6 P42226 1/20 0.79
CHEK1 O14757 1/20 0.79
HDAC3 O15379 1/20 0.79
ABCC4 O15439 1/20 0.79
GMNN O75496 1/20 0.79
LMNA P02545 1/20 0.79
CYP1A2 P05177 1/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydroxycamptothecin SCHEMBL28836816 1.00 TOP1 (0.98) TOP1MEN1KMT2ASMN1; SMN2ALDH1A1
Hydroxycamptothecin SCHEMBL9384413 0.99 TOP1 (1.00) TOP1MEN1KMT2ASMN1; SMN2ALDH1A1
Hydroxycamptothecin SCHEMBL25875 0.99 TOP1 (1.00) TOP1MEN1KMT2ASMN1; SMN2ALDH1A1
Hydroxycamptothecin SCHEMBL29929278 0.99 TOP1 (1.00) TOP1MEN1KMT2ASMN1; SMN2ALDH1A1
Hydroxycamptothecin SCHEMBL29350707 0.99 TOP1 (1.00) TOP1MEN1KMT2ASMN1; SMN2ALDH1A1
Hydroxycamptothecin SCHEMBL27638187 0.98 TOP1 (0.98) TOP1MEN1KMT2ASMN1; SMN2ALDH1A1
Hydroxycamptothecin SCHEMBL27905828 0.98 TOP1 (0.98) TOP1MEN1KMT2ASMN1; SMN2ALDH1A1
Hydroxycamptothecin SCHEMBL30872708 0.98 TOP1 (0.98) TOP1MEN1KMT2ASMN1; SMN2ALDH1A1
Hydroxycamptothecin SCHEMBL30426602 0.98 TOP1 (0.98) TOP1MEN1KMT2ASMN1; SMN2ALDH1A1
Hydroxycamptothecin SCHEMBL28094198 0.98 TOP1 (0.98) TOP1MEN1KMT2ASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101422156-A Agriculture bactericide composition and production method and use thereof UNIV ZHEJIANG FORESTRY (CN) 2009-05-06 CN claimed
CN-101243796-A Insecticide composition and its processing method UNIV ZHEJIANG FORESTRY (CN) 2008-08-20 CN claimed
CN-110859818-A Low-toxicity camptothecin nano-composite and preparation method and application thereof 河南省生物工程技术研究中心 2020-03-06 CN disclosed
CN-103432083-A Preparation process for glycyrrhizic acid-mediated hydroxycamptothecine albumin liver cancer targeting nanoparticle lyophilized powder UNIV NORTHEAST FORESTRY 2013-12-11 CN disclosed
CN-101654456-B Water-soluble derivants containing 10-hydroxycamptothecine and preparation method thereof MEDICAL RES INST CHONGQING UNIVERSITY OF MEDICAL SCIENCES 2013-01-23 CN disclosed
CN-1978448-B 10-hydroxy camptothecin arginine salt, and its preparing method and use CHENGDU SANKANG MEDICINE INST 2010-08-25 CN disclosed
CN-100592871-C Insecticide composition and its processing method UNIV ZHEJIANG FORESTRY 2010-03-03 CN disclosed
CN-101654456-A Water-soluble derivants containing 10-hydroxycamptothecine and preparation method thereof MEDICAL RES INST CHONGQING UNI 2010-02-24 CN disclosed
CN-101601642-A A kind of vesicle class drug-supplying system and application thereof UNIV SHENYANG PHARMACEUTICAL (CN) 2009-12-16 CN disclosed
CN-101422156-A Agriculture bactericide composition and production method and use thereof UNIV ZHEJIANG FORESTRY (CN) 2009-05-06 CN disclosed
CN-101243796-A Insecticide composition and its processing method UNIV ZHEJIANG FORESTRY (CN) 2008-08-20 CN disclosed
CN-1978447-A 10-hydroxy camptothecin arginine salt, and its preparing method and use CHENGDU SANKANG MEDICINE INST (CN) 2007-06-13 CN disclosed
CN-1978448-A 10-hydroxy camptothecin arginine salt, and its preparing method and use CHENGDU SANKANG MEDICINE INST (CN) 2007-06-13 CN disclosed
CN-1255104-C Camptothecine and hydroxy camptothecine lipid composition and its preparing method KANGHAI PHARMACEUTICAL CO LTD (CN) 2006-05-10 CN disclosed
CN-1554344-A Camptothecine and hydroxy camptothecine lipid composition and its preparing method 南京康海药业有限公司 2004-12-15 CN disclosed
CN-1167469-C Process for preparing nano particles of hydroxycamptothecine polylactate 黄石李时珍药业集团武汉李时珍药业有 2004-09-22 CN disclosed
CN-1158079-C Compound alkyl camptothecine injection prescription and prepn. process thereof 黄景健 2004-07-21 CN disclosed