SCHEMBL27469239

SCHEMBL27469239

c1ccc(C2CN(c3ccccc3)CCO2)cc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 1/20 0.51
LMNA P02545 1/20 0.50
ELOVL1 Q9BW60 2/20 0.47
CNR2 P34972 3/20 0.47
KDM4C Q9H3R0 1/20 0.47
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
GSK3B P49841 1/20 0.46
TSHR P16473 1/20 0.45
SYK P43405 1/20 0.44
NAPEPLD Q6IQ20 1/20 0.42
BPTF Q12830 1/20 0.42
FFAR2 O15552 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27469238 1.00 NUDT1 (0.51) NUDT1LMNAELOVL1CNR2KDM4C
SCHEMBL17602059 0.89 NUDT1 (0.46) NUDT1LMNAELOVL1CNR2KDM4C
SCHEMBL17602133 0.81 CNR2 (0.50) NUDT1ELOVL1CNR2KDM4CTSHR
SCHEMBL10785544 0.79 PDE10A (0.50) NUDT1CNR2KDM4CCYP1A2CYP2D6
SCHEMBL23379678 0.79 NUDT1 (0.52) NUDT1ELOVL1CNR2CYP1A2CYP2D6
SCHEMBL19888013 0.79 KDM4E (0.50) CNR2
SCHEMBL17602290 0.78 KDM4C (0.54) NUDT1ELOVL1CNR2KDM4CCYP1A2
SCHEMBL3794499 0.78 CNR2 (0.49) NUDT1CNR2SYK
SCHEMBL27559614 0.78 NUDT1 (0.54) NUDT1ELOVL1CYP1A2CYP2D6GSK3B
SCHEMBL8664503 0.78 SMN1; SMN2 (0.49) NUDT1LMNATSHRBPTF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1075812-C Prodrugs of morpholine tachykinin receptor antagonists MERCK & CO INC (US) 2001-12-05 CN disclosed
CN-1147254-A Prodrugs of morpholine tachykinin receptor antagonists MERCK & CO INC (US) 1997-04-09 CN disclosed