SCHEMBL8664503

SCHEMBL8664503

c1ccc(N2CCOC(c3cccs3)C2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.49
MAPT P10636 3/20 0.49
DRD4 P21917 1/20 0.42
DRD3 P35462 1/20 0.42
LMNA P02545 3/20 0.42
SLC6A9 P48067 1/20 0.42
RAB9A P51151 3/20 0.39
XBP1 P17861 1/20 0.39
KDM4E B2RXH2 1/20 0.37
TSHR P16473 1/20 0.37
HTT P42858 1/20 0.37
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36
BPTF Q12830 1/20 0.36
NOTUM Q6P988 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8665479 0.85 NPC1 (0.46) SMN1; SMN2MAPTLMNARAB9AKDM4E
SCHEMBL8997933 0.79 MAPT (0.32) SMN1; SMN2MAPTSLC6A9KDM4ETSHR
SCHEMBL27469239 0.78 NUDT1 (0.51) LMNATSHRBPTFNUDT1
SCHEMBL27469238 0.78 NUDT1 (0.51) LMNATSHRBPTFNUDT1
SCHEMBL18110505 0.77 SMN1; SMN2 (0.39) SMN1; SMN2MAPTLMNARAB9AXBP1
SCHEMBL30100998 0.76 CNR2 (0.53) DRD4DRD3
SCHEMBL30100985 0.75 BRD4 (0.40) SMN1; SMN2MAPTRAB9AKDM4ETSHR
SCHEMBL18110503 0.73 BRD4 (0.41) SMN1; SMN2MAPTRAB9AKDM4ETSHR
SCHEMBL19690771 0.71
SCHEMBL8917481 0.71 DRD3 (0.54) DRD4DRD3KDM4ETSHRHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852006-A N-aminoalkyl-substituted nitrogen-containing six membered heterocyclic compounds NIPPON CHEMIPHAR CO., LTD. (JP) 1998-12-22 US disclosed
US-5574030-A INHIBITING URINARY CONTRACTION, HETEROCYCLIC DIAMINES NIPPON CHEMIPHAR CO., LTD. (JP) 1996-11-12 US disclosed