SCHEMBL27469650

SCHEMBL27469650

COc1ccc(C(=O)c2ccccc2NC(=O)CN)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.59
ALDH1A1 P00352 5/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
KMT2A Q03164 3/20 0.54
MEN1 O00255 2/20 0.53
PKM P14618 2/20 0.53
F10 P00742 1/20 0.52
RAB9A P51151 3/20 0.51
MAPT P10636 2/20 0.51
USP2 O75604 1/20 0.51
TSHR P16473 1/20 0.51
GAA P10253 1/20 0.51
LMNA P02545 1/20 0.51
THRB P10828 1/20 0.51
NPC1 O15118 2/20 0.51
HDAC3 O15379 2/20 0.50
HDAC4 P56524 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL7622448 0.99 HCAR2 (0.57) HCAR2ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL11303046 0.84 ALDH1A1 (0.71) ALDH1A1KMT2AMEN1MAPTGAA
Bromide SCHEMBL7613349 0.83 ALDH1A1 (0.69) ALDH1A1KMT2AMEN1MAPTGAA
SCHEMBL9002518 0.81 F10 (0.72) ALDH1A1KMT2AMEN1PKMF10
SCHEMBL21129671 0.80 CYP1A2 (0.62) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL27455560 0.78 ALDH1A1 (0.52) ALDH1A1RAB9ANPC1HDAC3HDAC1
SCHEMBL19268078 0.78 KMT2A (0.54) HCAR2ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL12730395 0.78 KMT2A (0.78) ALDH1A1KMT2AMAPTTSHRGAA
SCHEMBL27457101 0.78 KMT2A (0.50) HCAR2ALDH1A1CYP1A2CYP2C19KMT2A
SCHEMBL7616103 0.78 NPSR1 (0.62) HCAR2ALDH1A1CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1145074-A Carbamoylmethylurea derivative SHIONOGI & CO (JP) 1997-03-12 CN disclosed