SCHEMBL7616103

SCHEMBL7616103

COc1ccc(C(=O)c2ccccc2NC(=O)CNC(=O)OCc2ccccc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 4/20 0.62
HTT P42858 4/20 0.62
LMNA P02545 1/20 0.62
ALDH1A1 P00352 8/20 0.51
HPGD P15428 2/20 0.51
HCAR2 Q8TDS4 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
MAPK1 P28482 1/20 0.48
RAF1 P04049 1/20 0.48
BRAF P15056 1/20 0.48
MAPT P10636 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
NPBWR1 P48145 1/20 0.47
MCHR1 Q99705 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
POLB P06746 1/20 0.47
CTDSP1 Q9GZU7 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7613630 0.90 NPSR1 (0.75) NPSR1HTTLMNAALDH1A1HPGD
SCHEMBL7617872 0.84 HTT (0.61) NPSR1HTTLMNAALDH1A1HPGD
SCHEMBL1484111 0.83 KDM4E (0.63) NPSR1HTTLMNAALDH1A1MEN1
SCHEMBL451742 0.81 LMNA (0.62) NPSR1HTTLMNAALDH1A1KMT2A
SCHEMBL7420731 0.80 KMT2A (0.59) NPSR1HTTLMNAALDH1A1MEN1
SCHEMBL9056505 0.80 NPC1 (0.57) LMNAALDH1A1MEN1KMT2AMAPT
SCHEMBL7611175 0.80 NPSR1 (0.58) NPSR1HTTLMNAALDH1A1HPGD
SCHEMBL27469650 0.78 HCAR2 (0.59) LMNAALDH1A1HCAR2MEN1KMT2A
SCHEMBL11785718 0.77 LMNA (0.77) NPSR1HTTLMNAALDH1A1MEN1
SCHEMBL7616469 0.77 HTT (0.55) NPSR1HTTLMNAALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0739903-B1 CARBAMOYLMETHYLUREA DERIVATIVE SHIONOGI & CO (JP) 2002-01-23 EP disclosed
US-5739162-A ANTAGONIST FOR GASTRIN AND/OR CHOLECYSTOKININ B-NOT A-RECEPTORS; SIDE EFFECT REDUCTION; ANTIULCER AGENTS; OPIOD-ENHANCING ANALGESICS; GASTROINTESTINAL DISORDERS; ANXIOLYTIC AGENTS SHIONOGI & CO., LTD. (JP) 1998-04-14 US disclosed
EP-0739903-A1 CARBAMOYLMETHYLUREA DERIVATIVE SHIONOGI & CO., LTD. (JP) 1996-10-30 EP disclosed