SCHEMBL27474353

SCHEMBL27474353

Cc1ccc2nc(Cl)nc(Cl)c2c1Cl

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 2/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
HTT P42858 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4167763 0.84 KDM4E (0.35) ALDH1A1KDM4ELMNAMAPTHTT
SCHEMBL3667600 0.79 HTT (0.32) HTTCYP3A4
SCHEMBL24815913 0.76 TNF (0.33) HTT
SCHEMBL29777989 0.76 ELANE (0.44) ALDH1A1KDM4E
SCHEMBL1997280 0.76 ELANE (0.44) ALDH1A1KDM4E
SCHEMBL27248807 0.76 PDE3B (0.40) ALDH1A1KDM4EMAPTPDE3BPDE3A
SCHEMBL27248775 0.72 TSHR (0.39) ALDH1A1KDM4EMAPT
SCHEMBL27248956 0.71 PDE3B (0.42) ALDH1A1KDM4EMAPTPDE3BPDE3A
SCHEMBL27474349 0.69 KDM4E (0.33) KDM4EMAPTPDE3BPDE3ACYP3A4
SCHEMBL27248563 0.68 ALDH1A1 (0.37) ALDH1A1KDM4EMAPTPDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12030857-B2 Glucose uptake inhibitors KADMON CORPORATION, LLC (US) 2024-07-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12030857-B2 Glucose uptake inhibitors SLC2A1, SLC2A4, SLC2A2 ALDH1A1 1422/4885KDM4E 2325/4885LMNA 4856/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.