SCHEMBL3667600

SCHEMBL3667600

Clc1nc(Cl)c2c(Cl)c(Cl)ccc2n1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.32
CYP2A6 P11509 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
CYP3A4 P08684 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28320224 0.79 HTT (0.37) HTT
SCHEMBL24815913 0.79 TNF (0.33) HTT
SCHEMBL27474353 0.79 ALDH1A1 (0.34) HTTCYP3A4
SCHEMBL27248775 0.75 TSHR (0.39) MAPK1
SCHEMBL27248807 0.75 PDE3B (0.40)
SCHEMBL27248563 0.75 ALDH1A1 (0.37)
SCHEMBL30013654 0.74 PARP1 (0.44) TDP1
SCHEMBL3337344 0.74 PARP1 (0.44) TDP1
SCHEMBL4167763 0.71 KDM4E (0.35) HTTCYP3A4MAPK1
SCHEMBL23577134 0.71 TNKS (0.33) HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102584721-B Synthetic method of 2,4-dichloroquinazoline derivative UNIV ZHEJIANG TECHNOLOGY 2014-07-02 CN disclosed
CN-103534251-A Novel compounds for organic electronic material and organic electroluminescent device using the same ROHM & HAAS ELECT MAT 2014-01-22 CN disclosed
CN-102584721-A Synthetic method of 2,4-dichloroquinazoline derivative UNIV ZHEJIANG TECHNOLOGY 2012-07-18 CN disclosed
EP-2238119-A1 QUINAZOLINES AND RELATED HETEROCYCLIC COMPOUNDS, AND THEIR THERAPEUTIC USE Vereniging voor Christelijk Hoger Onderwijs, Wetenschappelijk Onderzoek en Patiëntenzorg (NL) 2010-10-13 EP disclosed
WO-2009083608-A1 QUINAZOLINES AND RELATED HETEROCYCLIC COMPOUNDS, AND THEIR THERAPEUTIC USE VERENIGING VOOR CHRISTELIJK HOGER ONDERWIJS, WETENSCHAPPELIJK ONDERZOEK EN PATIENTENZORG (NL) 2009-07-09 WO disclosed
CN-1044245-C Tricyclic Dicarbonyl derivatives HAFFMANN LA ROCHE AG F (DE) 1999-07-21 CN disclosed
CN-1149295-A Tricyclic Dicarbonyl derivatives HOFFMANN LA ROCHE (CH) 1997-05-07 CN disclosed