SCHEMBL27475990

SCHEMBL27475990

NCc1cccc(N2CCNCC2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 7/20 0.60
HTR1A P08908 6/20 0.60
ADRB1 P08588 4/20 0.57
HTR3E A5X5Y0 4/20 0.57
HTR3B O95264 4/20 0.57
HTR3A P46098 4/20 0.57
HTR3D Q70Z44 4/20 0.57
HTR3C Q8WXA8 4/20 0.57
SIGMAR1 Q99720 4/20 0.57
HTR2C P28335 3/20 0.57
THRB P10828 2/20 0.57
HTR6 P50406 2/20 0.57
TP53 P04637 1/20 0.57
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
HTR2A P28223 1/20 0.57
SLC6A4 P31645 1/20 0.57
CYP2C19 P33261 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27483822 0.98 HTR7 (0.58) HTR7HTR1AADRB1HTR3EHTR3B
Piperazine SCHEMBL28850703 0.98 HTR7 (0.58) HTR7HTR1AADRB1HTR3EHTR3B
Hydrochloric Acid SCHEMBL27355289 0.98 HTR7 (0.58) HTR7HTR1AADRB1HTR3EHTR3B
SCHEMBL28323356 0.91 HTR7 (0.50) HTR7HTR1AADRB1HTR3EHTR3B
SCHEMBL27662780 0.87 AGXT (0.56) SIGMAR1DRD2DRD3ALDH1A1MAPT
SCHEMBL109316 0.84 AGXT (0.67) ALDH1A1MAPTAGXT
SCHEMBL27581488 0.83 ADRB1 (0.48) HTR7HTR1AADRB1HTR3EHTR3B
SCHEMBL301359 0.83 ADRB1 (0.62) HTR7HTR1AADRB1HTR3EHTR3B
SCHEMBL3204004 0.83 HTR7 (0.60) HTR7HTR1AADRB1HTR3EHTR3B
SCHEMBL7415117 0.83 HTR7 (0.62) HTR7HTR1AADRB1HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 75 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110452130-A A kind of Obovatol Mannich base analog derivative and the preparation method and application thereof UNIV SHANXI AGRICULTURAL 2019-11-15 CN claimed
CN-110437191-A 13- amino Xanthatin analog derivative and its preparation method and application UNIV SHANXI AGRICULTURAL 2019-11-12 CN claimed
CN-110337293-A Therapeutic compound 新泽西鲁特格斯州立大学 2019-10-15 CN claimed
CN-106699690-A Pleuromulin derivative with acyl piperazine side chain and preparing method and application of pleuromulin derivative 华南农业大学 2017-05-24 CN claimed
CN-104507950-B Thienopyrimidines 拜耳医药股份有限公司 2017-03-22 CN claimed
CN-102797043-B Medicinal molecular fragment library and construction process thereof Tianli (Tianjin) Technology Co., Ltd. (CN) 2015-11-25 CN claimed
CN-102797043-A Medicinal molecular fragment library and construction method thereof CBB NETWORK CO LTD 2012-11-28 CN claimed
CN-106420754-B The purposes of benzo five-membered Azacyclyl bridged piperazine derivatives 沈阳海王生物技术有限公司 2019-11-05 CN disclosed
CN-110354267-A Method and composition for low blood pressure recovery 法尔麦兹公司 2019-10-22 CN disclosed
CN-110337293-A Therapeutic compound 新泽西鲁特格斯州立大学 2019-10-15 CN disclosed
CN-107573302-B Aryl piperazines compound and its preparation method and application 袁牧 2019-09-20 CN disclosed
CN-106699690-B A kind of pleuromutilin derivative and its preparation method and application with acyl piperazine base side chain 华南农业大学 2019-09-10 CN disclosed
CN-104926801-B Substituted azetidine analog derivative, the pharmaceutical composition containing it and its application in antitumor 浙江大学 2019-06-04 CN disclosed
CN-1145609-C Piperazine compounds and medical use thereof ������ҩ��ʽ���� 2004-04-14 CN disclosed
CN-1306526-A Novel heterocyclically substituted amides with cysteine protease-inhibiting effect BASF AG (DE) 2001-08-01 CN disclosed
CN-1281438-A Piperazine compounds and their use as pharmaceuticals EFUKU CO LTD (JP) 2001-01-24 CN disclosed
CN-1271363-A 3' -N-modified 6-O-substituted erythromycin ketolide derivatives having antibacterial activity ABBOTT LAB (US) 2000-10-25 CN disclosed
CN-1261347-A Remedies/preventives for frequent urination/urinary incontinence and tropone derivatives NIPPON KAYAKU KK (JP) 2000-07-26 CN disclosed
CN-1237183-A 6-0-substituted ketolides with antibacterial activity ABBOTT CO (US) 1999-12-01 CN disclosed
CN-1224427-A 6-O-substituted erythromycin compounds and preparation method thereof ABBOTT LAB (US) 1999-07-28 CN disclosed