SCHEMBL27486372

SCHEMBL27486372

CN(C)C(c1ccc(C#N)cc1)C1CCCCC1(O)C(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 18/20 0.53
TSHR P16473 1/20 0.38
ESR1 P03372 1/20 0.35
PGR P06401 1/20 0.35
HTR2A P28223 1/20 0.35
SLC6A3 Q01959 1/20 0.35
TRPC5 Q9UL62 1/20 0.35
HSD11B1 P28845 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6936758 0.81 SLC6A4 (0.40) TRPA1TSHRSLC6A3HSD11B1
SCHEMBL5160386 0.67 OPRM1 (0.44) SLC6A3HSD11B1
SCHEMBL6939057 0.65 SLC6A4 (0.42) TRPA1SLC6A3HSD11B1
SCHEMBL6939750 0.65 TSHR (0.42) TSHRHSD11B1
SCHEMBL5163207 0.64 OPRM1 (0.44) SLC6A3
SCHEMBL5159940 0.64 OPRM1 (0.40) TSHRSLC6A3
SCHEMBL5158046 0.63 OPRM1 (0.43) TRPA1TSHRSLC6A3
SCHEMBL6938861 0.62 GRIN2B (0.39) TRPA1
SCHEMBL5158611 0.62 OPRM1 (0.41) TRPA1SLC6A3
SCHEMBL7732583 0.61 OPRM1 (0.38) TSHRSLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1183098-C 3-amino-3-aryl-1-alcohol derivatives and preparation and use thereof 2005-01-05 CN claimed
CN-1270162-A 3-amino-3-aryl-1-alcohol derivatives and preparation and use thereof GRUENENTHAL GMBH (DE) 2000-10-18 CN claimed
CN-1183098-C 3-amino-3-aryl-1-alcohol derivatives and preparation and use thereof 2005-01-05 CN disclosed
CN-1270162-A 3-amino-3-aryl-1-alcohol derivatives and preparation and use thereof GRUENENTHAL GMBH (DE) 2000-10-18 CN disclosed