SCHEMBL27488013

SCHEMBL27488013

CC(Cc1ccc(F)cc1)CC(N)C(C)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.44
TRPA1 O75762 1/20 0.42
CPA1 P15085 1/20 0.42
TPH1 P17752 2/20 0.40
REN P00797 2/20 0.40
PPARG P37231 2/20 0.40
PPARA Q07869 2/20 0.40
MAPK1 P28482 1/20 0.40
SLC7A5 Q01650 1/20 0.39
PTGS1 P23219 3/20 0.38
PTGS2 P35354 3/20 0.38
LMNA P02545 2/20 0.38
CYP2C9 P11712 2/20 0.38
AKR1C3 P42330 2/20 0.38
CXCR1 P25024 2/20 0.38
CXCR2 P25025 2/20 0.38
ALB P02768 1/20 0.38
ESR1 P03372 1/20 0.38
ALOX5 P09917 1/20 0.38
RARB P10826 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27488010 0.86 ALPI (0.53) RENSLC7A5PTGS1
SCHEMBL27505422 0.85 DPP4 (0.42) KMT2AMAPK1PTGS1PTGS2ALDH1A1
SCHEMBL27506207 0.85 SLC6A2 (0.50) RENPPARGPPARALMNACYP2C9
SCHEMBL27505438 0.83 SLC1A1 (0.57) KMT2ARENPPARGPPARASLC7A5
SCHEMBL4989923 0.79 MME (0.43) KMT2ATRPA1CPA1PPARGPPARA
SCHEMBL27507830 0.77 PPARG (0.42) PPARGPPARAALDH1A1
SCHEMBL8587665 0.75 ENPEP (0.47) KMT2ATRPA1CPA1TPH1PPARA
SCHEMBL27506589 0.74 TRPA1 (0.47) KMT2ATRPA1CPA1PPARGPPARA
SCHEMBL5794436 0.74 TRPA1 (0.50) KMT2ATRPA1CPA1CYP2C9
SCHEMBL1913524 0.74 CACNA2D1 (0.50) KMT2ATRPA1CPA1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101862317-A The pregabalin derivant that is used for the treatment of fibromyalgia and other disease WARNER LAMBERT CO 2010-10-20 CN disclosed
CN-1310872-C Mono- and disubstituted 3-propyl gamma-aminobutyric acids WARNER LAMBERT CO (US) 2007-04-18 CN disclosed
CN-1726023-A Pregabalin derivatives for the treatment of fibromyalgia and other diseases WARNER LAMBERT CO (US) 2006-01-25 CN disclosed
CN-1660779-A Mono- and disubstituted 3-propyl gamma-aminobutyric acids WARNER LAMBERT CO (US) 2005-08-31 CN disclosed
CN-1625393-A Alpha 2 delta ligands to treat tinnitus WARNER LAMBERT CO (US) 2005-06-08 CN disclosed
CN-1196671-C Mono-and disubstituted 3-propyl-gamma-aminobutyric acids WARNER LAMBERT CO (US) 2005-04-13 CN disclosed
CN-1355784-A Mono-and disubstituted 3-propyl-gamma-aminobutyric acids WARNER LAMBERT CO (US) 2002-06-26 CN disclosed