SCHEMBL27488187

SCHEMBL27488187

COC(=O)[C@@H](N)Cc1ccc(-c2cn(C)c(=O)cc2C)cc1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.42
DPP7 Q9UHL4 2/20 0.42
ALDH1A1 P00352 1/20 0.41
BRD4 O60885 4/20 0.40
TPH1 P17752 2/20 0.38
ITGA4 P13612 1/20 0.38
ITGB7 P26010 1/20 0.38
BAZ2B Q9UIF8 1/20 0.36
BAZ2A Q9UIF9 1/20 0.36
PTGS2 P35354 1/20 0.36
SCN9A Q15858 1/20 0.36
TYR P14679 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27488188 1.00 DPP4 (0.42) DPP4DPP7ALDH1A1BRD4TPH1
SCHEMBL5163064 0.80 ITGA4 (0.39) ALDH1A1BRD4TPH1ITGA4ITGB7
SCHEMBL6236587 0.79 ITGB1 (0.41) ALDH1A1TPH1ITGA4PTGS2
Hydrochloric Acid SCHEMBL5165900 0.79 ALDH1A1 (0.41) ALDH1A1TPH1ITGA4ITGB7PTGS2
Hydrochloric Acid SCHEMBL6236581 0.78 ALDH1A1 (0.42) ALDH1A1TPH1ITGA4PTGS2
SCHEMBL6238973 0.78 ALDH1A1 (0.40) ALDH1A1TPH1ITGA4ITGB7PTGS2
Hydrochloric Acid SCHEMBL27502521 0.78 ALDH1A1 (0.42) ALDH1A1TPH1ITGA4PTGS2
SCHEMBL27487456 0.78 ALDH1A1 (0.40) ALDH1A1TPH1ITGA4ITGB7PTGS2
Hydrochloric Acid SCHEMBL6239874 0.77 ALDH1A1 (0.42) ALDH1A1TPH1ITGA4ITGB7PTGS2
Hydrochloric Acid SCHEMBL27487816 0.77 ALDH1A1 (0.42) ALDH1A1TPH1ITGA4ITGB7PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1196682-C 4-pyridyl-N-acyl-L-phenylalanine HOFFMANN LA ROCHE (CH) 2005-04-13 CN disclosed
CN-1402709-A 4-pyridinyl-N-acyl-L-phenylalanines HOFFMANN LA ROCHE (CH) 2003-03-12 CN disclosed