SCHEMBL27489451

SCHEMBL27489451

[c]1cc2ccccc2cc1-c1ncc[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 6/20 0.46
NISCH Q9Y2I1 2/20 0.46
MTOR P42345 1/20 0.46
ADK P55263 1/20 0.46
ADRA2B P18089 5/20 0.39
ADRA2C P18825 5/20 0.39
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CSNK1A1 P48729 1/20 0.36
TYRO3 Q06418 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP19A1 P11511 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
IDO1 P14902 1/20 0.36
KCNK13 Q9HB14 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9404099 0.74 ADRA2A (0.44) ADRA2ANISCHMTORADKADRA2B
SCHEMBL4719727 0.74 ADRA2A (0.44) ADRA2ANISCHMTORADKADRA2B
SCHEMBL6163163 0.73 CYP2A6 (0.37) ALDH1A1MEN1KMT2ACYP1A2CYP3A4
SCHEMBL295727 0.72 NISCH (0.52) ADRA2ANISCHMTORADKADRA2B
SCHEMBL703704 0.71 NISCH (0.47) ADRA2ANISCHMTORADKADRA2B
SCHEMBL7391931 0.71 NISCH (0.56) ADRA2ANISCHMTORADKADRA2B
SCHEMBL2093036 0.71 MTOR (0.44) ADRA2ANISCHMTORADKADRA2B
SCHEMBL29613953 0.70 NISCH (0.60) ADRA2ANISCHMTORADKADRA2B
SCHEMBL4329170 0.70 ADRA2A (0.50) ADRA2ANISCHMTORADKADRA2B
SCHEMBL534893 0.70 NISCH (0.60) ADRA2ANISCHMTORADKADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100398555-C Protease inhibitors for coronaviruses and SARS-COV and the use thereof CYTOVIA INC (US) 2008-07-02 CN disclosed
CN-1235875-C Substituted alpha-hydroxy acid caspase inhibitors and uses thereof CYTOVIA INC (US) 2006-01-11 CN disclosed
CN-1176941-C Caspase inhibitors and the use thereof ά 2004-11-24 CN disclosed
CN-1382119-A Substituted alpha-hydroxy acid caspase inhibitors and uses thereof CYTOVIA INC (US) 2002-11-27 CN disclosed
CN-1349496-A Caspase inhibitors and uses thereof CYTOVIA INC (US) 2002-05-15 CN disclosed
CN-1346344-A Substituted 2-aminobenzamide caspase ihibitors and the use thereof CYTOVIA INC (US) 2002-04-24 CN disclosed