SCHEMBL27490347

SCHEMBL27490347

CCCCn1cncc1-c1cccnc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 1/20 0.51
CYP2A6 P11509 4/20 0.47
ALDH1A1 P00352 2/20 0.47
CYP2A13 Q16696 1/20 0.47
CYP2C9 P11712 5/20 0.47
CYP2C19 P33261 5/20 0.47
CYP3A4 P08684 5/20 0.47
CYP2D6 P10635 2/20 0.47
CYP19A1 P11511 1/20 0.47
CYP1A2 P05177 3/20 0.44
HK1 P19367 1/20 0.44
HKDC1 Q2TB90 1/20 0.44
HIF1A Q16665 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CNR2 P34972 1/20 0.44
ICMT O60725 1/20 0.44
CYP2E1 P05181 2/20 0.43
CYP2B6 P20813 2/20 0.43
CYP11B1 P15538 5/20 0.43
CYP11B2 P19099 5/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL593796 0.86 CYP11B1 (0.58) TLR8ALDH1A1CNR2CYP11B1CYP11B2
SCHEMBL1502180 0.78 IDO1 (0.49) ICMTCYP11B1CYP11B2IDO1
SCHEMBL27984310 0.78 CYP11B1 (0.51) TLR8ALDH1A1CYP2C19CYP1A2CNR2
SCHEMBL7683890 0.78 CYP2A6 (0.43) TLR8CYP2A6ALDH1A1CYP2A13CYP2C9
SCHEMBL10983627 0.77 IDO1 (0.44) ALDH1A1CYP3A4HIF1AHSD17B10CYP11B1
SCHEMBL15653534 0.77 CYP11B1 (0.54) TLR8ALDH1A1CNR2CYP11B1CYP11B2
SCHEMBL20409162 0.77 ADORA2A (0.38) TLR8ALDH1A1ICMTCYP11B1CYP11B2
SCHEMBL1502091 0.76 CYP11B1 (0.62) ALDH1A1CYP3A4CYP2D6CYP1A2CYP11B1
SCHEMBL31627317 0.75 CYP2A6 (0.62) CYP2A6ALDH1A1CYP2A13CYP2C9CYP2C19
SCHEMBL1133225 0.75 CYP2A6 (0.62) CYP2A6ALDH1A1CYP2A13CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1211385-C Bicyclic imidazo-5-yl-amine derivs. GRUENENTHAL GMBH (DE) 2005-07-20 CN disclosed
CN-1402726-A Bicyclic imidazo-5-yl-amine derivs. GRUENENTHAL GMBH (DE) 2003-03-12 CN disclosed