SCHEMBL27499643

SCHEMBL27499643

CC(C(=O)C(C)c1cnc(-c2ccccc2)s1)c1cnc(-c2ccccc2)s1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 8/20 0.50
ALDH1A1 P00352 7/20 0.50
NPC1 O15118 7/20 0.50
RAB9A P51151 7/20 0.50
MAPT P10636 5/20 0.50
HDAC1 Q13547 2/20 0.48
HDAC6 Q9UBN7 1/20 0.48
CCNE1 P24864 5/20 0.45
CDK2 P24941 5/20 0.45
CDK5 Q00535 5/20 0.45
CCNT1 O60563 1/20 0.45
CDK1 P06493 1/20 0.45
CDK4 P11802 1/20 0.45
CCNB1 P14635 1/20 0.45
CCNA2 P20248 1/20 0.45
CCND1 P24385 1/20 0.45
CDK7 P50613 1/20 0.45
CDK9 P50750 1/20 0.45
CCNH P51946 1/20 0.45
MNAT1 P51948 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12790160 0.81 ALDH1A1 (0.46) SMN1; SMN2ALDH1A1NPC1RAB9AMAPT
SCHEMBL2819462 0.81 ALDH1A1 (0.47) SMN1; SMN2ALDH1A1NPC1RAB9AMAPT
SCHEMBL27769540 0.81 PDE2A (0.43) SMN1; SMN2ALDH1A1NPC1RAB9AMAPT
SCHEMBL20558976 0.78 NPC1 (0.44) SMN1; SMN2ALDH1A1NPC1RAB9AMAPT
SCHEMBL2199263 0.78 NPC1 (0.44) SMN1; SMN2ALDH1A1NPC1RAB9AMAPT
SCHEMBL7040603 0.77 ALDH1A1 (0.43) SMN1; SMN2ALDH1A1NPC1RAB9AMAPT
SCHEMBL27688647 0.77 KDM4E (0.43) SMN1; SMN2ALDH1A1NPC1RAB9AMAPT
SCHEMBL10153257 0.75 NPC1 (0.42) SMN1; SMN2ALDH1A1NPC1RAB9AMAPT
SCHEMBL10191826 0.75 ALDH1A1 (0.42) SMN1; SMN2ALDH1A1NPC1RAB9AMAPT
SCHEMBL12788371 0.75 NPC1 (0.46) SMN1; SMN2ALDH1A1NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1230166-C Gyrase inhibitors and uses thereof VERTEX PHARMA (US) 2005-12-07 CN disclosed
CN-1400898-A Gyrase inhibitors and uses thereof VERTEX PHARMA (US) 2003-03-05 CN disclosed