SCHEMBL27500466

SCHEMBL27500466

NC(=O)N(c1ccccc1Br)c1ccccc1NS(=O)(=O)c1cc(Cl)sc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACLY P53396 1/20 0.48
CYP2C9 P11712 1/20 0.46
S100A9 P06702 3/20 0.45
TDP1 Q9NUW8 1/20 0.44
CDK1 P06493 2/20 0.41
CCNB1 P14635 2/20 0.41
CCNA2 P20248 2/20 0.41
CCND1 P24385 2/20 0.41
CDK2 P24941 2/20 0.41
CDK7 P50613 2/20 0.41
CCNH P51946 2/20 0.41
CCNA1 P78396 2/20 0.41
CDK6 Q00534 2/20 0.41
PFKFB3 Q16875 1/20 0.41
PIK3C3 Q8NEB9 1/20 0.41
PTGES2 Q9H7Z7 2/20 0.38
SGK1 O00141 1/20 0.37
IDH1 O75874 1/20 0.37
MCL1 Q07820 1/20 0.36
APP P05067 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27566179 0.83 PTGES2 (0.57) ACLYPFKFB3PTGES2
SCHEMBL7552185 0.79 ACLY (0.53) ACLYCYP2C9S100A9TDP1CDK1
SCHEMBL27498931 0.78 KMT2A (0.43) ACLY
SCHEMBL27576135 0.78 MCL1 (0.46) MCL1
SCHEMBL27535606 0.76 MEN1 (0.54) CYP2C9MCL1
SCHEMBL7593518 0.76 ACLY (0.61) ACLYCYP2C9S100A9TDP1CDK1
SCHEMBL27575358 0.75 MEN1 (0.45) ACLYTDP1PTGES2
SCHEMBL27517617 0.75 PKM (0.47) PTGES2
SCHEMBL27516979 0.73 GAA (0.57) TDP1
SCHEMBL7589357 0.72 S100A9 (0.57) ACLYCYP2C9S100A9TDP1CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1539816-A IL-8 receptor antagonists ʷ��˿�������ȳ�ķ���޹�˾ 2004-10-27 CN disclosed
CN-1355697-A IL-8 receptor antagonists SMITHKLINE BEECHAM CORP (US) 2002-06-26 CN disclosed
CN-1215990-A IL-8 receptor antagonists SMITHKLINE BEECHAM CORP (US) 1999-05-05 CN disclosed