SCHEMBL27516632

SCHEMBL27516632

O=C(C(Cc1ccc(F)cc1)c1cccc(F)c1)C(Cc1ccc(F)cc1)c1cccc(F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
CNR2 P34972 1/20 0.46
CES2 O00748 1/20 0.45
CES1 P23141 1/20 0.45
SLC6A9 P48067 1/20 0.45
SLC6A5 Q9Y345 1/20 0.45
PPARA Q07869 2/20 0.43
PPARG P37231 1/20 0.43
EPHX1 P07099 2/20 0.41
SLC1A1 P43005 2/20 0.41
KCNQ2 O43526 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
PPARD Q03181 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27608061 0.80 MDM2 (0.48) HDAC4HDAC7HDAC5CNR2CES2
SCHEMBL29609176 0.80 EPHX1 (0.71) HDAC4HDAC7HDAC5CNR2PPARA
SCHEMBL28107951 0.80 EPHX1 (0.71) HDAC4HDAC7HDAC5CNR2PPARA
SCHEMBL27586693 0.79 HDAC4 (0.49) HDAC4HDAC7HDAC5CNR2CES2
SCHEMBL27991442 0.77 EPHX1 (0.58) CNR2PPARAPPARGEPHX1
SCHEMBL27695771 0.76 NR3C2 (0.42) PPARAPPARD
SCHEMBL3374627 0.76 CNR1 (0.53) HDAC4HDAC7HDAC5CNR2PPARA
SCHEMBL5178070 0.76 EPHX1 (0.49) CNR2EPHX1
SCHEMBL4664796 0.76 PPARA (0.56) PPARAPPARGEPHX1PPARDTDP1
SCHEMBL27516633 0.75 CNR2 (0.38) HDAC4HDAC7HDAC5CNR2CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1951939-A Novel pyrrole derivatives as pharmaceutical agents LILLY CO ELI (US) 2007-04-25 CN disclosed
CN-1269820-C Novel pyrrole derivatives as medicaments LILLY CO ELI (US) 2006-08-16 CN disclosed
CN-1511157-A Novel pyrrole derivatives as medicaments 2004-07-07 CN disclosed