SCHEMBL27543607

SCHEMBL27543607

CC(C)(C)OOC(=O)c1cccc(CBr)c1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.58
TSHR P16473 1/20 0.58
HSD17B10 Q99714 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
SLC7A5 Q01650 3/20 0.46
LOXL2 Q9Y4K0 1/20 0.45
CYP4F2 P78329 4/20 0.44
CYP4A11 Q02928 4/20 0.44
MEP1B Q16820 1/20 0.41
MRGPRX4 Q96LA9 2/20 0.39
FOLH1 Q04609 1/20 0.38
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27960544 0.88 ALDH1A1 (0.55) ALDH1A1TSHRHSD17B10TDP1SLC7A5
SCHEMBL27796426 0.85 LOXL2 (0.65) ALDH1A1TSHRHSD17B10TDP1SLC7A5
SCHEMBL27775507 0.85 ALDH1A1 (0.58) ALDH1A1TSHRHSD17B10TDP1SLC7A5
SCHEMBL127411 0.84 SLC7A5 (0.62) SLC7A5LOXL2CYP4F2CYP4A11MEP1B
SCHEMBL29471996 0.84 SLC7A5 (0.62) SLC7A5LOXL2CYP4F2CYP4A11MEP1B
SCHEMBL27476536 0.84 ALDH1A1 (0.54) ALDH1A1TSHRHSD17B10TDP1SLC7A5
SCHEMBL224130 0.84 ALDH1A1 (0.75) ALDH1A1TSHRHSD17B10TDP1SLC7A5
SCHEMBL27960526 0.82 ALDH1A1 (0.55) ALDH1A1TSHRHSD17B10TDP1SLC7A5
SCHEMBL28528856 0.81 ALDH1A1 (0.54) ALDH1A1TSHRHSD17B10TDP1SLC7A5
SCHEMBL27571589 0.81 ALDH1A1 (0.61) ALDH1A1TSHRHSD17B10TDP1LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109952297-A Compound 奥斯陆大学 2019-06-28 CN disclosed
CN-103052636-B D 2antagonist and synthetic method thereof and using method Altos Therapeutics, LLC (US) 2016-03-09 CN disclosed
CN-103052636-A D2 antagonists, methods of synthesis and methods of use ALTOS THERAPEUTICS LLC 2013-04-17 CN disclosed
CN-1261276-A Protease inhibitors SMITHKLINE BEECHAM CORP (US) 2000-07-26 CN disclosed