SCHEMBL27545274

SCHEMBL27545274

COc1ccc(C(=O)c2nn[nH]c2C(=O)O)cc1OC

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
CA12 O43570 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA4 P22748 1/20 0.54
CA6 P23280 1/20 0.54
CA7 P43166 1/20 0.54
TPMT P51580 1/20 0.54
CA9 Q16790 1/20 0.54
CA14 Q9ULX7 1/20 0.54
GAA P10253 2/20 0.51
APAF1 O14727 1/20 0.49
NSD2 O96028 1/20 0.49
CASP3 P42574 1/20 0.49
SENP8 Q96LD8 1/20 0.49
SENP7 Q9BQF6 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27480820 0.89 TSHR (0.55) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL5165358 0.84 CYP2C19 (0.49) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL5515197 0.83 TSHR (0.54) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL27552756 0.80 CYP1A2 (0.44) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL5167917 0.80 CYP2C19 (0.50) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL4770528 0.75 PDE4A (0.50) CA12CA1CA2CA4CA6
SCHEMBL5516179 0.74 CYP1A2 (0.43) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL1493250 0.74 CYP1A2 (1.00) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6872165 0.73 TSHR (0.81) TSHRCYP1A2CYP3A4CYP2C9CYP2C19
Veratric Acid SCHEMBL976032 0.72 CA12 (1.00) TSHRCYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1312135-C Tricyclic triazolobenzazepine * derivatives, process for preparing the same, and antiallergic agent MEIJI SEIKA KAISHA (JP) 2007-04-25 CN disclosed