SCHEMBL27550522

SCHEMBL27550522

O=C1NC(=O)C(c2ccccc2N2CCCCC2)C(=O)N1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.46
NPC1 O15118 1/20 0.44
EEF2K O00418 1/20 0.43
MAPK1 P28482 2/20 0.41
ALDH1A1 P00352 5/20 0.40
MAPT P10636 3/20 0.40
GAA P10253 2/20 0.40
KDM4E B2RXH2 2/20 0.40
L3MBTL1 Q9Y468 3/20 0.40
EGFR P00533 1/20 0.40
RAF1 P04049 1/20 0.40
ALOX12 P18054 1/20 0.40
MAP2K1 Q02750 1/20 0.40
KCNQ2 O43526 1/20 0.39
TSHR P16473 2/20 0.37
PRKDC P78527 1/20 0.37
OPRM1 P35372 1/20 0.36
OPRK1 P41145 1/20 0.36
OPRL1 P41146 1/20 0.36
HTR1A P08908 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30442171 0.74 CRBN (0.57) EEF2KALDH1A1TSHROPRM1
SCHEMBL23064465 0.71 KEAP1 (0.52) KEAP1NPC1EEF2KMAPK1ALDH1A1
SCHEMBL8704351 0.71 EEF2K (0.46) KEAP1NPC1EEF2KMAPK1ALDH1A1
SCHEMBL23064544 0.69 PDCD1 (0.51) KEAP1NPC1EEF2KMAPK1GAA
SCHEMBL29559516 0.69 SMN1; SMN2 (0.56) KEAP1NPC1EEF2KMAPK1ALDH1A1
SCHEMBL27934132 0.69 MAPK1 (0.74) KEAP1NPC1MAPK1ALDH1A1MAPT
SCHEMBL23064483 0.69 KEAP1 (0.48) KEAP1NPC1EEF2KMAPK1ALDH1A1
SCHEMBL11876685 0.69 IDO1 (0.37) ALDH1A1MAPTGAAKDM4EL3MBTL1
SCHEMBL31198346 0.69 KEAP1 (0.48) KEAP1NPC1EEF2KMAPK1ALDH1A1
SCHEMBL18701462 0.68 HTR2C (0.50) KEAP1MAPK1HTR1AADRA1BHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1318406-C New barbituric acid derivatives, processes for their prodn. and pharmaceutical agent contg. same BOEHRINGER MANNHEIM GMBH (DE) 2007-05-30 CN disclosed