SCHEMBL27560331

SCHEMBL27560331

C=CCCCCN(C(N)=O)c1ccc2[nH]cc(C3CCN(CCCCC)CC3)c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 4/20 0.44
HTR1D P28221 7/20 0.44
HTR1B P28222 6/20 0.44
DRD2 P14416 4/20 0.44
CHRM2 P08172 1/20 0.44
MAPT P10636 1/20 0.42
BLM P54132 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
SLC6A4 P31645 1/20 0.42
HTR2A P28223 5/20 0.42
HTR7 P34969 5/20 0.42
HTR1A P08908 1/20 0.42
HTR2C P28335 1/20 0.42
HTR1E P28566 1/20 0.42
HTR1F P30939 1/20 0.42
DRD3 P35462 1/20 0.42
HTR2B P41595 1/20 0.42
HTR6 P50406 1/20 0.42
CCR5 P51681 1/20 0.42
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27483636 0.89 HTR1D (0.48) HTR1DHTR1BDRD2CHRM2SLC6A4
SCHEMBL8707969 0.84 DRD2 (0.42) CCR2DRD2SLC6A4HTR1ADRD3
SCHEMBL8707108 0.81 SLC6A4 (0.43) HTR1DHTR1BMAPTBLMNPSR1
SCHEMBL27527184 0.81 HTR1D (0.50) CCR2HTR1DHTR1BDRD2CHRM2
SCHEMBL7479525 0.78 HTR1D (0.48) CCR2HTR1DHTR1BDRD2CHRM2
SCHEMBL7481757 0.77 HTR1D (0.55) HTR1DHTR1BDRD2CHRM2HTR1A
SCHEMBL7487120 0.77 CCR2 (0.61) CCR2HTR1DHTR1BDRD2CHRM2
SCHEMBL27498570 0.75 HTR1D (0.51) CCR2HTR1DHTR1BDRD2CHRM2
SCHEMBL27498200 0.75 HTR1D (0.49) HTR1DHTR1BDRD2CHRM2HTR2A
SCHEMBL27496223 0.75 HTR1D (0.65) HTR1DHTR1BDRD2CHRM2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1184425-A 5-substituted-3- (1,2,3, 6-tetrahydropyridin-4-yl) -and 3- (piperidin-4-yl) -1H-indoles, 5-HT1FAgonists LILLY CO ELI (US) 1998-06-10 CN disclosed